SCHEMBL9613974

SCHEMBL9613974

O=C(O)C(CCCCCCc1ccccc1)S(=O)(=O)CCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.48
MAPT P10636 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
S1PR2 O95136 1/20 0.43
S1PR4 O95977 1/20 0.43
S1PR1 P21453 1/20 0.43
S1PR3 Q99500 1/20 0.43
HDAC1 Q13547 3/20 0.43
HDAC2 Q92769 2/20 0.43
CA2 P00918 1/20 0.43
ALOX5 P09917 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
LTB4R Q15722 1/20 0.42
GRIK1 P39086 1/20 0.42
HDAC3 O15379 1/20 0.42
MAPK1 P28482 1/20 0.42
ADRA1A P35348 1/20 0.42
HDAC4 P56524 1/20 0.42
SLC6A3 Q01959 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10420392 1.00 TRPA1 (0.48) TRPA1MAPTRXFP1S1PR2S1PR4
SCHEMBL9614055 0.94 TRPA1 (0.48) TRPA1MAPTRXFP1S1PR2S1PR4
SCHEMBL9614242 0.92 TDP1 (0.43) TRPA1MAPTRXFP1S1PR2S1PR1
SCHEMBL9858450 0.92 PPARA (0.48) TRPA1MAPTRXFP1HDAC1HDAC2
SCHEMBL9614107 0.92 PPARA (0.48) TRPA1MAPTRXFP1HDAC1HDAC2
SCHEMBL9614112 0.92 PPARA (0.48) TRPA1MAPTRXFP1HDAC1HDAC2
SCHEMBL27272794 0.92 TRPA1 (0.42) TRPA1MAPTRXFP1S1PR2S1PR4
SCHEMBL9857963 0.90 ALDH1A1 (0.44) TRPA1MAPTHDAC1TRPV1
SCHEMBL9613963 0.89 TRPA1 (0.49) TRPA1MAPTRXFP1S1PR2S1PR4
SCHEMBL9614317 0.89 MMP3 (0.52) ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5145611-A Diabetes BOEHRINGER MANNHEIM GMBH (DE) 1992-09-08 US claimed
US-5145611-A Diabetes BOEHRINGER MANNHEIM GMBH (DE) 1992-09-08 US disclosed
EP-0279162-B1 CARBONIC ACID DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICALS CONTAINING THEM Roche Diagnostics GmbH (DE) 1991-06-19 EP disclosed
EP-0279162-A1 Carbonic acid derivatives, process for their preparation and pharmaceuticals containing them Roche Diagnostics GmbH (DE) 1988-08-24 EP disclosed