SCHEMBL9615085

SCHEMBL9615085

COC(=O)c1ccc(C(=O)NC(CSC(C)=O)Cc2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 1/20 0.51
PIN1 Q13526 2/20 0.49
CTSL P07711 1/20 0.48
RAB9A P51151 3/20 0.48
NPC1 O15118 2/20 0.48
MAPK1 P28482 2/20 0.46
ROCK2 O75116 1/20 0.46
RPS6KA5 O75582 1/20 0.46
RPS6KA4 O75676 1/20 0.46
PRKACA P17612 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
IRAK1 P51617 1/20 0.46
PRKX P51817 1/20 0.46
ROCK1 Q13464 1/20 0.46
PRKG1 Q13976 1/20 0.46
PKN2 Q16513 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
SGK2 Q9HBY8 1/20 0.46
CYP3A4 P08684 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9459542 0.85 MAPT (0.45) RAB9ANPC1MAPK1CYP3A4CYP1A2
SCHEMBL8837469 0.80 FCER2 (0.50) CTRB1RAB9ANPC1MAPK1CYP3A4
SCHEMBL9588793 0.79 CYP3A4 (0.46) RAB9ANPC1MAPK1CYP3A4CYP1A2
SCHEMBL7450894 0.78 MME (0.52) RAB9ANPC1MAPK1CYP3A4CYP1A2
SCHEMBL9587602 0.77 MME (0.48) CTRB1RAB9ANPC1MAPK1CYP3A4
SCHEMBL9068533 0.77 MME (0.62) MAPK1CYP3A4MME
SCHEMBL18576675 0.76 CTRB1 (0.65) CTRB1CTSLCYP3A4CYP1A2CYP2C9
SCHEMBL9588619 0.76 CYP3A4 (0.54) CTRB1RAB9ANPC1MAPK1CYP3A4
SCHEMBL9587952 0.76 MME (0.47) CTRB1RAB9ANPC1MAPK1CYP3A4
SCHEMBL9459027 0.75 SLC7A5 (0.42) RAB9AALDH1A1SLC7A5MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4112865-A None JP disclosed
JP-H04112865-A SUBSTITUTED AMIDE DERIVATIVE DAINIPPON PHARMACEUT CO LTD 1992-04-14 JP disclosed