SCHEMBL9616628

SCHEMBL9616628

Nc1ccccc1NS(=O)(=O)c1c(Cl)ccc2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.44
SLC40A1 Q9NP59 5/20 0.44
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MCL1 Q07820 1/20 0.41
MAPK14 Q16539 1/20 0.41
NFKBIA P25963 2/20 0.40
RELA Q04206 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
KEAP1 Q14145 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
METAP2 P50579 1/20 0.39
METAP1 P53582 1/20 0.39
CYP2A6 P11509 1/20 0.39
HDAC1 Q13547 1/20 0.38
HTR1A P08908 1/20 0.38
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9616784 0.77 HTR6 (0.54) HSP90AA1HSP90AB1MEN1KMT2AALDH1A1
SCHEMBL9616674 0.77 HSP90AA1 (0.49) HSP90AA1HSP90AB1MEN1KMT2AMCL1
SCHEMBL9616556 0.77 MEN1 (0.56) SLC40A1MEN1KMT2AMCL1ALDH1A1
SCHEMBL9616814 0.75 BRD4 (0.42) RECQLSLC40A1MEN1KMT2AALDH1A1
SCHEMBL9616695 0.74 HSP90AA1 (0.47) HSP90AA1HSP90AB1MEN1KMT2AALDH1A1
SCHEMBL8416358 0.73 CYP2A6 (0.50) HSP90AA1HSP90AB1MEN1KMT2AALDH1A1
SCHEMBL30737433 0.72 PTGES2 (0.56) SLC40A1MEN1KMT2AMCL1NFKBIA
SCHEMBL9616615 0.72 MEN1 (0.61) HSP90AA1HSP90AB1MEN1KMT2AMAPT
SCHEMBL4191121 0.72 PTGES2 (0.69) MEN1KMT2AALDH1A1MAPTPTGES2
SCHEMBL499404 0.71 CYP2A6 (0.52) MEN1KMT2AALDH1A1MAPTKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462179-A4 NOVEL SULFONAMIDES AS RADIOSENSITIZERS 1992-03-18 EP claimed
EP-0462179-A1 NOVEL SULFONAMIDES AS RADIOSENSITIZERS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-12-27 EP claimed
WO-1990009787-A1 NOVEL SULFONAMIDES AS RADIOSENSITIZERS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1990-09-07 WO claimed