SCHEMBL9621782

SCHEMBL9621782

Nc1cccc(C(=O)O)c1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
KDM4E B2RXH2 1/20 0.54
HPGD P15428 1/20 0.54
HSD17B10 Q99714 1/20 0.54
PTGS1 P23219 1/20 0.50
CNR2 P34972 1/20 0.50
ADORA1 P30542 1/20 0.49
KMO O15229 2/20 0.47
RORB Q92753 3/20 0.46
RORC P51449 2/20 0.46
KIF11 P52732 1/20 0.46
TRPM2 O94759 1/20 0.46
PARP1 P09874 2/20 0.45
GRIK1 P39086 1/20 0.45
IKBKB O14920 1/20 0.45
BRD4 O60885 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
XDH P47989 1/20 0.44
MEN1 O00255 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6801907 0.85 RXRA (0.51) ALDH1A1KDM4EHPGDHSD17B10CNR2
SCHEMBL17744870 0.84 MMP2 (0.55) ALDH1A1KDM4EHPGDHSD17B10KMO
SCHEMBL30086172 0.84 MMP2 (0.55) ALDH1A1KDM4EHPGDHSD17B10KMO
SCHEMBL30279482 0.81 KDM4E (0.64) ALDH1A1KDM4EHPGDHSD17B10PTGS1
SCHEMBL22497505 0.81 KDM4E (0.64) ALDH1A1KDM4EHPGDHSD17B10PTGS1
SCHEMBL9188681 0.80 MCL1 (0.57) ALDH1A1KDM4EHPGDHSD17B10PARP1
SCHEMBL2935772 0.80 CNR2 (0.52) ALDH1A1PTGS1CNR2ADORA1KIF11
SCHEMBL10588475 0.79 RORB (0.56) ALDH1A1KDM4EHPGDHSD17B10ADORA1
SCHEMBL4077919 0.79 MMP2 (0.57) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL4724483 0.78 PARP1 (0.59) ALDH1A1KDM4ECNR2ADORA1RORB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0182569-B1 Use of 1,6-dimethyl-4-oxo-1,6,7,8,9a-hexahydro-4H-pyrido[1,2-a]pyrimidine-3-carboxamide for the prevention and treatment of gastrointestinal damages CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1992-01-29 EP disclosed