SCHEMBL9622227

SCHEMBL9622227

FNc1ccc(C(F)(F)F)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.54
EPHX2 P34913 1/20 0.54
CA1 P00915 2/20 0.50
CA2 P00918 1/20 0.50
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
CA12 O43570 1/20 0.45
MMP2 P08253 1/20 0.45
TGM2 P21980 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
PTGS1 P23219 2/20 0.42
TRPV1 Q8NER1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921455 0.80 EPHX2 (0.56) KIF11EPHX2CA1CA2ALDH1A1
SCHEMBL394422 0.80 EPHX2 (0.56) KIF11EPHX2CA1CA2ALDH1A1
SCHEMBL7267375 0.79 KIF11 (0.50) KIF11EPHX2CA1CA2ALDH1A1
SCHEMBL63468 0.78 ALDH1A1 (0.67) KIF11EPHX2ALDH1A1TSHR
SCHEMBL1776928 0.76 KIF11 (0.52) KIF11EPHX2CA1CA2ALDH1A1
SCHEMBL11023642 0.76 EPHX2 (0.58) KIF11EPHX2CA1CA2CA12
SCHEMBL9725672 0.76 KIF11 (0.52) KIF11EPHX2CA1CA2ALDH1A1
SCHEMBL14674966 0.76 KIF11 (0.52) KIF11EPHX2CA1CA2ALDH1A1
SCHEMBL378918 0.76 CA1 (0.54) KIF11EPHX2CA1CA2ALDH1A1
SCHEMBL27764151 0.76 KIF11 (0.52) KIF11EPHX2CA1CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110305045-A A kind of amides compound and its purposes in treating cancer 成都海创药业有限公司 2019-10-08 CN disclosed
CN-105622580-B Benzimidazole as prolyl hydroxylase inhibitors 詹森药业有限公司 2019-06-21 CN disclosed
CN-109071518-A Oxazoline vacation dimer, medical composition and its use 普渡制药公司 2018-12-21 CN disclosed
CN-102026985-B Quinazoline derivatives as RAF kinase modulators and methods and uses thereof 埃姆比特生物科学公司 2016-07-06 CN disclosed
CN-105622580-A Benzoimidazoles as prolyl hydroxylase inhibitors JANSSEN PHARMACEUTICA NV 2016-06-01 CN disclosed
CN-102076680-B Benzimidazoles as Prolyl Hydroxylase Inhibitors JANSSEN PHARMACEUTICA N.V. (BE) 2016-03-02 CN disclosed
CN-102119156-B Substituted pyrroles and methods of use GENENTECH INC 2015-01-21 CN disclosed
CN-101927187-B Catalyst for oligomerization and polymerization of ethylene and preparation method and application thereof CHINA PETROLEUM & CHEMICAL 2012-07-04 CN disclosed
CN-102076694-A 5, 6, 7, 8-tetrahydro-imidazo[1, 5-a]pyrazine compounds ACTELION PHARMACEUTICALS LTD 2011-05-25 CN disclosed
CN-101440090-B 2-(6'-imine pyridinyl) benzoxazole metal complexes, as well as preparation method and application thereof CHINESE ACAD INST CHEMISTRY 2011-01-26 CN disclosed
CN-101927187-A Catalyst for oligomerization and polymerization of ethylene and preparation method and application thereof CHINA PETROLEUM & CHEMICAL 2010-12-29 CN disclosed
CN-101440090-A 2-(6'-imine pyridinyl) benzoxazole metal complexes, as well as preparation method and application thereof CHINESE ACAD INST CHEMISTRY (CN) 2009-05-27 CN disclosed
CN-1227548-A Substituted p-trifluoromethylphenyluracils BAYER AG (DE) 1999-09-01 CN disclosed
US-5096928-A Caterpillars BAYER AKTIENGESELLSCHAFT (DE) 1992-03-17 US disclosed