SCHEMBL9725672

SCHEMBL9725672

FC(F)(F)c1ccc(NS)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.52
EPHX2 P34913 1/20 0.52
CA1 P00915 2/20 0.48
CA2 P00918 1/20 0.48
CA12 O43570 1/20 0.44
MMP2 P08253 1/20 0.44
TGM2 P21980 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
PTGS1 P23219 2/20 0.41
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921455 0.78 EPHX2 (0.56) KIF11EPHX2CA1CA2RAB9A
SCHEMBL394422 0.78 EPHX2 (0.56) KIF11EPHX2CA1CA2RAB9A
SCHEMBL63468 0.76 ALDH1A1 (0.67) KIF11EPHX2ALDH1A1TSHR
SCHEMBL9622227 0.76 KIF11 (0.54) KIF11EPHX2CA1CA2CA12
SCHEMBL378918 0.74 CA1 (0.54) KIF11EPHX2CA1CA2CA12
SCHEMBL11023642 0.74 EPHX2 (0.58) KIF11EPHX2CA1CA2CA12
SCHEMBL1776928 0.74 KIF11 (0.52) KIF11EPHX2CA1CA2CA12
SCHEMBL16274236 0.74 MAPT (0.45)
SCHEMBL14674966 0.74 KIF11 (0.52) KIF11EPHX2CA1CA2CA12
SCHEMBL12364124 0.74 TSHR (0.48) KIF11EPHX2CA1CA2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022268145-A1 AMIDE COMPOUND, AND PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF 中国科学院上海药物研究所 2022-12-29 WO disclosed
CN-115504940-A Amide compound, preparation method and pharmaceutical application thereof 中国科学院上海药物研究所 2022-12-23 CN disclosed
CN-101265224-B Method for preparing 4-trifluoromethylmercaptoaniline JINTAN LINGYUN CHEMICAL FACTORY 2010-12-08 CN disclosed
US-5095032-A PARASITICIDAL NEW SUBSTITUTED THIENOPYRANONES BAYER AKTIENGESELLSCHAFT (DE) 1992-03-10 US disclosed
US-4804655-A Pesticidal cyclic malonylphosphonic diamides BAYER AKTIENGESELLSCHAFT (DE) 1989-02-14 US disclosed
US-4771048-A VETERINARY MEDICINE BAYER AKTIENGESELLSCHAFT (DE) 1988-09-13 US disclosed
US-4766144-A 3-carbamoyl-4-hydroxy-coumarins for combating parasitic heiminths BAYER AKTIENGESELLSCHAFT (DE) 1988-08-23 US disclosed
US-4459304-A MITICIDES, NEMATOCIDES, FUNGICIDES, BACTERICIDES, INSECTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1984-07-10 US disclosed
US-4318919-A Combating bacteria with tetrachlorophthalamic acids BAYER AKTIENGESELLSCHAFT (DE) 1982-03-09 US disclosed
US-4277499-A Combating insects with N-(substituted-phenyl)-N-(2-chloro-6-fluoro-benzoyl)-ureas BAYER AKTIENGESELLSCHAFT (DE) 1981-07-07 US disclosed
US-4276310-A ARTHROPODICIDES, FUNGICIDES, BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1981-06-30 US disclosed