SCHEMBL9623846

SCHEMBL9623846

C[C@H]1C[C@@H]2C(=CC[C@@]3(C)[C@H]2CC[C@]3(O)C#N)[C@@]2(C)C=CC(=O)C=C12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
KCNH2 Q12809 1/20 0.42
CYP19A1 P11511 6/20 0.40
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
CYP3A4 P08684 5/20 0.37
HIF1A Q16665 4/20 0.37
NR3C1 P04150 4/20 0.37
PGR P06401 4/20 0.37
NR1I2 O75469 2/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
LMNA P02545 1/20 0.37
CYP2C9 P11712 1/20 0.37
ABCB11 O95342 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ABCC4 O15439 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12265813 0.86 NFKB1 (0.46) NFKB1NFKB2RELAKCNH2CYP19A1
SCHEMBL9623669 0.82 NFKB1 (0.56) NFKB1NFKB2RELAKCNH2CYP19A1
SCHEMBL13069741 0.82 HIF1A (0.52) NFKB1NFKB2RELAKCNH2CYP19A1
SCHEMBL3394762 0.82 HIF1A (0.52) NFKB1NFKB2RELAKCNH2CYP19A1
SCHEMBL9073247 0.80 HIF1A (0.55) NFKB1NFKB2RELAKCNH2FNTA
SCHEMBL12266195 0.80 HIF1A (0.55) NFKB1NFKB2RELAKCNH2FNTA
SCHEMBL8859711 0.80 HIF1A (0.55) NFKB1NFKB2RELAKCNH2FNTA
SCHEMBL15144388 0.80 NFKB1 (0.47) NFKB1NFKB2RELAKCNH2CYP19A1
SCHEMBL17549314 0.80 NFKB1 (0.46) NFKB1NFKB2RELAKCNH2CYP19A1
SCHEMBL9624281 0.80 NR3C1 (0.43) CYP19A1CYP3A4HIF1ANR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268400-B1 STEROIDAL 17ALPHA-SILYL ETHERS AND PROCESS TO CORTICOIDS AND PROGESTERONES THE UPJOHN COMPANY (US) 1992-04-29 EP claimed