SCHEMBL9624550

SCHEMBL9624550

COc1ccc2c(c1OC)CCN(CCCN(C)CCc1c[nH]c3c(C)cccc13)C2=O

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.42
MAPT P10636 2/20 0.42
HCN4 Q9Y3Q4 1/20 0.42
CNR2 P34972 1/20 0.41
ALOX15 P16050 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 1/20 0.41
CYP3A4 P08684 1/20 0.41
SMPD1 P17405 1/20 0.37
DRD2 P14416 2/20 0.37
DRD4 P21917 2/20 0.37
DRD3 P35462 1/20 0.37
HTR2A P28223 2/20 0.36
ABCB1 P08183 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HTR4 Q13639 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624815 0.86 KDM4E (0.45) HTR6MAPTHCN4ALOX15KDM4E
SCHEMBL9624930 0.85 MAPT (0.42) HTR6MAPTHCN4CNR2ALOX15
SCHEMBL9624754 0.84 HTR1A (0.47) HTR6MAPTHCN4NPC1RAB9A
SCHEMBL9624987 0.83 SLC6A4 (0.49) MAPTHCN4CNR2ALOX15CYP3A4
SCHEMBL9624107 0.82 MAPT (0.42) MAPTHCN4CNR2ALOX15CYP3A4
SCHEMBL9624988 0.81 MAPT (0.42) MAPTHCN4CNR2ALOX15CYP3A4
SCHEMBL10645652 0.81 HCN4 (0.63) HTR6MAPTHCN4ALOX15KDM4E
SCHEMBL9624887 0.80 HTR6 (0.45) HTR6MAPTHCN4ALOX15CYP3A4
SCHEMBL9624614 0.80 HTR1D (0.51) HTR6MAPTHCN4CNR2KDM4E
SCHEMBL9624011 0.80 HCN4 (0.46) MAPTHCN4CNR2ALOX15KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed