SCHEMBL9624754

SCHEMBL9624754

COc1ccc2[nH]cc(CCN(C)CCCN3CCc4c(ccc(OC)c4OC)C3=O)c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.47
HTR2A P28223 3/20 0.47
HTR6 P50406 2/20 0.47
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
HTR1D P28221 1/20 0.47
HTR1B P28222 1/20 0.47
HTR2C P28335 1/20 0.47
HTR1E P28566 1/20 0.47
HTR1F P30939 1/20 0.47
HTR7 P34969 1/20 0.47
HTR2B P41595 1/20 0.47
HTR3A P46098 1/20 0.47
HTR5A P47898 1/20 0.47
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47
HTR4 Q13639 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624930 0.92 MAPT (0.42) HTR1AHTR2AHTR6HTR3EHTR3B
SCHEMBL9624987 0.91 SLC6A4 (0.49) HTR1AKMT2AMAPTMEN1LMNA
SCHEMBL9624614 0.91 HTR1D (0.51) HTR6HTR1DKMT2AMAPTMEN1
SCHEMBL9624308 0.88 HTR1A (0.48) HTR1AHTR2AHTR6HTR3EHTR3B
SCHEMBL9624855 0.84 HCN4 (0.44) HTR1AMTNR1AMTNR1BMAPTSLC6A4
SCHEMBL9624550 0.84 HTR6 (0.42) HTR2AHTR6HTR4MAPTSMN1; SMN2
SCHEMBL9623770 0.82 MAPT (0.42) HTR1AKMT2AMAPTMEN1SMN1; SMN2
SCHEMBL9624225 0.82 HCN4 (0.44) HTR1AMAPTSLC6A4HCN4
SCHEMBL10649533 0.82 HCN4 (0.62) HTR1AHTR2AHTR6HTR3EHTR3B
SCHEMBL9624897 0.82 HTR1A (0.52) HTR1AHTR2AHTR6HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed