(Cyclopentylamino)Methylenediphosphonic Acid

(Cyclopentylamino)Methylenediphosphonic Acid

SCHEMBL9626232

O=P(O)(O)C(NC1CCCC1)P(=O)(O)O

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 3/20 0.46
ERAP2 Q6P179 3/20 0.46
MMP2 P08253 7/20 0.45
CA12 O43570 5/20 0.45
CA1 P00915 5/20 0.45
CA2 P00918 5/20 0.45
CA9 Q16790 5/20 0.45
MMP1 P03956 2/20 0.45
MMP8 P22894 2/20 0.43
MMP3 P08254 1/20 0.43
FDPS P14324 1/20 0.39
EPHX1 P07099 5/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPT P10636 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Incadronic Acid SCHEMBL223885 0.98 ANPEP (0.48) ANPEPERAP2MMP2CA12CA1
(Cyclohexylamino)Methylenediphosphonic Acid SCHEMBL8370913 0.98 ANPEP (0.48) ANPEPERAP2MMP2CA12CA1
(Cyclooctylamino)Methylenediphosphonic Acid SCHEMBL9777403 0.98 ANPEP (0.48) ANPEPERAP2MMP2CA12CA1
(Cyclobutylamino)Methylenediphosphonic Acid SCHEMBL9626988 0.95 MMP2 (0.45) ANPEPERAP2MMP2CA12CA1
Incadronic Acid SCHEMBL2898450 0.94 ANPEP (0.46) ANPEPERAP2MMP2CA12CA1
(Cyclopropylamino)Methylenediphosphonic Acid SCHEMBL9627717 0.90 MMP2 (0.41) ANPEPERAP2MMP2CA12CA1
Incadronic Acid SCHEMBL2898447 0.82 ANPEP (0.41) ANPEPERAP2MMP2CA12CA1
SCHEMBL9627714 0.80 MMP2 (0.39) ANPEPERAP2MMP2CA12CA1
SCHEMBL9777781 0.80 FDPS (0.41) ANPEPERAP2MMP2MMP8FDPS
SCHEMBL10419330 0.80 HDAC3 (0.33) ANPEPERAP2MMP2MMP1MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325482-B1 (CYCLOALKYLAMINO)METHYLENEBISPHOSPHONIC ACIDS AND MEDICINES CONTAINING THEM YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1992-04-01 EP disclosed
US-5041428-A Bone resorption inhibitor, antiarthritic agent YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1991-08-20 US disclosed
US-4970335-A ANTIARTHRITIC AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1990-11-13 US disclosed
EP-0325482-A1 (Cycloalkylamino)methylenebisphosphonic acids and medicines containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1989-07-26 EP disclosed