SCHEMBL9627248

SCHEMBL9627248

CC(=O)[C@@]1(O)[C@H](C)C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)CC[C@]4(C)C3=CC[C@@]21C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
TSHR P16473 2/20 0.50
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
KCNH2 Q12809 1/20 0.42
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
NR3C1 P04150 4/20 0.41
HIF1A Q16665 3/20 0.38
LMNA P02545 3/20 0.38
MEN1 O00255 2/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP2C19 P33261 1/20 0.38
CYP19A1 P11511 3/20 0.38
AR P10275 5/20 0.37
SERPINA6 P08185 2/20 0.35
CYP3A4 P08684 3/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8203795 0.92 NFKB1 (0.44) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL10623020 0.90 ALDH1A1 (0.54) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL8470203 0.89 NFKB1 (0.46) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL8470202 0.89 NFKB1 (0.46) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL10419014 0.89 NFKB1 (0.54) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL9619163 0.89 NFKB1 (0.54) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL8207710 0.89 NFKB1 (0.54) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL8192700 0.89 NFKB1 (0.54) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL3083179 0.89 NFKB1 (0.54) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL7565596 0.89 NFKB1 (0.54) ALDH1A1TSHRNFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276393-B1 PROCESS FOR THE PREPARATION OF 6-ALPHA, 9-ALPHA-DIFLUORO-11-BETA-17-ALPHA-DIHYDROXY-16-ALPHA-METHYL-PREGN-4-ENE-3,20-DIONE AND ITS DERIVATIVES SCHERING AKTIENGESELLSCHAFT (DE) 1992-03-04 EP claimed
US-4898693-A Process for production of 6α,9α-difluoro-11β,17α-dihydroxy-16α-methyl-4-pregnene-3,20-dione and its derivatives SCHERING AKTIENGESELLSCHAFT (DE) 1990-02-06 US claimed
EP-0276393-A2 Process for the preparation of 6-alpha, 9-alpha-difluoro-11-beta-17-alpha-dihydroxy-16-alpha-methyl-pregn-4-ene-3,20-dione and its derivatives SCHERING AKTIENGESELLSCHAFT (DE) 1988-08-03 EP claimed
EP-0276393-B1 PROCESS FOR THE PREPARATION OF 6-ALPHA, 9-ALPHA-DIFLUORO-11-BETA-17-ALPHA-DIHYDROXY-16-ALPHA-METHYL-PREGN-4-ENE-3,20-DIONE AND ITS DERIVATIVES SCHERING AKTIENGESELLSCHAFT (DE) 1992-03-04 EP disclosed
US-4898693-A Process for production of 6α,9α-difluoro-11β,17α-dihydroxy-16α-methyl-4-pregnene-3,20-dione and its derivatives SCHERING AKTIENGESELLSCHAFT (DE) 1990-02-06 US disclosed
EP-0276393-A2 Process for the preparation of 6-alpha, 9-alpha-difluoro-11-beta-17-alpha-dihydroxy-16-alpha-methyl-pregn-4-ene-3,20-dione and its derivatives SCHERING AKTIENGESELLSCHAFT (DE) 1988-08-03 EP disclosed