SCHEMBL9627910

SCHEMBL9627910

CCCN(CCC)CC1COc2ccc(OC)cc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.44
DRD2 P14416 3/20 0.44
HTR2A P28223 3/20 0.44
HTR2C P28335 3/20 0.44
DRD1 P21728 1/20 0.44
HTR1B P28222 1/20 0.44
HTR2B P41595 2/20 0.44
SIGMAR1 Q99720 2/20 0.44
DRD3 P35462 2/20 0.42
HTR7 P34969 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
CYP3A4 P08684 3/20 0.40
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9628688 0.88 HTR2B (0.43) HTR1ADRD2HTR2AHTR2CHTR2B
SCHEMBL24090506 0.82 HTR2B (0.55) HTR1ADRD2HTR2BSIGMAR1DRD3
SCHEMBL9406456 0.81 HTR1D (0.44) HTR1ADRD2DRD1HTR1BDRD3
SCHEMBL9627777 0.81 PPARG (0.37) HTR1ADRD2HTR2AHTR2CDRD1
SCHEMBL9627835 0.81 DRD3 (0.46) DRD2DRD3CYP3A4ALDH1A1TP53
Methylamine SCHEMBL10700891 0.80 HTR1A (0.50) HTR1ADRD2HTR2CHTR2BSIGMAR1
SCHEMBL9628089 0.79 ACHE (0.41) CYP3A4KMT2A
SCHEMBL9628958 0.78 PPARG (0.39) HTR1AHTR2C
SCHEMBL9262060 0.78 MTNR1A (0.53) HTR1ADRD2HTR2AHTR2CDRD1
SCHEMBL9627798 0.77 HTR1A (0.50) HTR1ADRD2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP disclosed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP disclosed