SCHEMBL9628146

SCHEMBL9628146

CCCN(CCC)CC1CCc2ccc(OC(=O)c3c(F)cccc3F)cc21

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACHE P22303 10/20 0.45
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
NQO2 P16083 4/20 0.40
MTNR1A P48039 4/20 0.40
MTNR1B P49286 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9629884 0.90 ACHE (0.45) ACHENQO2MTNR1AMTNR1B
SCHEMBL9627778 0.85 MCHR1 (0.48) ACHEADRA2AADRA2BADRA2CADRA1D
SCHEMBL9627883 0.82 ACHE (0.45) ACHENQO2MTNR1AMTNR1B
SCHEMBL10458915 0.81 KMT2A (0.45) ACHE
SCHEMBL9628081 0.81 ACHE (0.60) ACHE
SCHEMBL9628479 0.80 ACHE (0.44) ACHENQO2MTNR1AMTNR1B
SCHEMBL9628568 0.80 PTGS2 (0.43) ACHENQO2MTNR1AMTNR1B
SCHEMBL9628113 0.77 MTNR1A (0.53) NQO2MTNR1AMTNR1B
SCHEMBL9628591 0.73 ACHE (0.47) ACHENQO2MTNR1AMTNR1B
SCHEMBL9628952 0.73 ACHE (0.66) ACHENQO2MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP disclosed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP disclosed