SCHEMBL9630604

SCHEMBL9630604

CCCc1sc(-c2ccccc2)nc1OC(=O)c1ccccc1

nearest known ligand 0.77

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 5/20 0.72
KDM4E B2RXH2 1/20 0.57
MEN1 O00255 1/20 0.57
ALDH1A1 P00352 1/20 0.57
KMT2A Q03164 1/20 0.57
NLRP1 Q9C000 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.51
RARA P10276 1/20 0.47
RARB P10826 1/20 0.47
RARG P13631 1/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.46
TRPM8 Q7Z2W7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9629413 0.87 ALOX5 (0.75) ALOX5L3MBTL1TRPM8
SCHEMBL9630227 0.84 ALOX5 (1.00) ALOX5L3MBTL1RARARARBRARG
SCHEMBL9628650 0.84 ALOX5 (1.00) ALOX5MEN1ALDH1A1KMT2AL3MBTL1
SCHEMBL9628625 0.81 ALOX5 (0.78) ALOX5KMT2AL3MBTL1TRPM8
SCHEMBL9629268 0.81 ALOX5 (0.77) ALOX5L3MBTL1TRPM8
SCHEMBL9630562 0.80 ALOX5 (0.66) ALOX5L3MBTL1TRPM8
SCHEMBL9629404 0.73 TRPM8 (0.59) ALOX5TRPM8
SCHEMBL7693031 0.71 ALOX5 (0.57) ALOX5
SCHEMBL15049221 0.69 MEN1 (0.63) ALOX5KDM4EMEN1ALDH1A1KMT2A
SCHEMBL27412605 0.68 KDM4E (0.59) ALOX5KDM4EMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5124342-A Antiinflammatory, antiarthritic agents; antiallergens; skin disorders ABBOTT LABORATORIES (US) 1992-06-23 US disclosed
EP-0457803-A4 4-HYDROXYTHIAZOLES AS 5-LIPOXYGENASE INHIBITORS 1991-12-04 EP disclosed
EP-0457803-A1 4-HYDROXYTHIAZOLES AS 5-LIPOXYGENASE INHIBITORS ABBOTT LABORATORIES (US) 1991-11-27 EP disclosed
WO-1990009801-A1 4-HYDROXYTHIAZOLES AS 5-LIPOXYGENASE INHIBITORS ABBOTT LABORATORIES (US) 1990-09-07 WO disclosed
WO-1990009381-A1 4-HYDROXYTHIAZOLES AS 5-LIPOXYGENASE INHIBITORS ABBOTT LABORATORIES (US) 1990-08-23 WO disclosed