SCHEMBL9632

SCHEMBL9632

CCOC(=O)CCc1ccc(-c2ccccc2)c(-c2onc(C)c2N)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
CYP4F2 P78329 2/20 0.43
CYP4A11 Q02928 2/20 0.43
PTPN1 P18031 5/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 2/20 0.39
HPGD P15428 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
P2RY12 Q9H244 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
FAAH O00519 1/20 0.37
NPC1 O15118 1/20 0.36
PKM P14618 1/20 0.36
NFKB1 P19838 1/20 0.36
RAB9A P51151 1/20 0.36
NFKB2 Q00653 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4663 0.80 CYP4F2 (0.51) ALDH1A1CYP4F2CYP4A11KDM4EHPGD
SCHEMBL9973 0.80 SYK (0.38) ALDH1A1CYP4F2CYP4A11PTPN1SMN1; SMN2
SCHEMBL9631 0.78 PTGS1 (0.40) ALDH1A1SMN1; SMN2KDM4EHPGDL3MBTL1
Hydrochloric Acid SCHEMBL27782843 0.78 CYP4F2 (0.54) ALDH1A1CYP4F2CYP4A11PTPN1SMN1; SMN2
SCHEMBL15822278 0.72 ALOX5 (0.51) ALDH1A1CYP4F2CYP4A11PTPN1SMN1; SMN2
SCHEMBL15823568 0.72 ALOX5 (0.51) ALDH1A1CYP4F2CYP4A11PTPN1SMN1; SMN2
SCHEMBL3744 0.71 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2KDM4EL3MBTL1MAPT
SCHEMBL2772418 0.70 CYP4F2 (0.68) CYP4F2CYP4A11PTPN1
SCHEMBL9633 0.70 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2KDM4EHPGDL3MBTL1
SCHEMBL8903063 0.70 TDP1 (0.56) CYP4F2CYP4A11PTPN1APPSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed