SCHEMBL9633

SCHEMBL9633

CCOC(=O)C(C)c1ccc(-c2ccccc2-c2onc(C)c2N)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
KDM4E B2RXH2 3/20 0.39
KMT2A Q03164 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 2/20 0.39
MEN1 O00255 2/20 0.39
APAF1 O14727 2/20 0.39
USP2 O75604 2/20 0.39
POLB P06746 2/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PKM P14618 2/20 0.37
LPAR1 Q92633 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9631 0.88 PTGS1 (0.40) ALDH1A1SMN1; SMN2KDM4EKMT2AL3MBTL1
SCHEMBL9974 0.77 LPAR1 (0.40) ALDH1A1SMN1; SMN2KDM4EKMT2AL3MBTL1
SCHEMBL27915165 0.74 TSHR (0.43) ALDH1A1SMN1; SMN2KDM4ELMNAHPGD
SCHEMBL6188617 0.73 GRIA4 (0.50) ALDH1A1KMT2AL3MBTL1LMNAMEN1
SCHEMBL13653511 0.72 AKR1C3 (0.50) ALDH1A1SMN1; SMN2KDM4EKMT2AL3MBTL1
SCHEMBL7358 0.70 LPAR1 (0.40) ALDH1A1SMN1; SMN2KMT2AL3MBTL1MEN1
SCHEMBL9632 0.70 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2KDM4EL3MBTL1MAPT
SCHEMBL1625348 0.69 LMNA (0.55) ALDH1A1SMN1; SMN2KDM4EKMT2ALMNA
Methylamine SCHEMBL11586903 0.69 MMP8 (0.54) SMN1; SMN2KMT2ALMNAMEN1NPC1
SCHEMBL10756249 0.69 MMP8 (0.57) SMN1; SMN2KMT2ALMNAMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed