SCHEMBL9632764

SCHEMBL9632764

COC(=O)c1nccnc1C(C)=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.52
L3MBTL1 Q9Y468 2/20 0.50
KDM4E B2RXH2 7/20 0.44
ALDH1A1 P00352 4/20 0.38
KDM4C Q9H3R0 2/20 0.38
MAPK1 P28482 2/20 0.38
KDM6B O15054 1/20 0.38
KDM5C P41229 1/20 0.38
KDM2A Q9Y2K7 1/20 0.38
KDM3A Q9Y4C1 1/20 0.38
STAT3 P40763 1/20 0.38
HIF1A Q16665 1/20 0.38
TSHR P16473 2/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
DYRK1A Q13627 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL71518 0.93 NPSR1 (0.59) NPSR1L3MBTL1KDM4EALDH1A1KDM4C
SCHEMBL24994251 0.85 NPSR1 (0.46) NPSR1L3MBTL1KDM4EALDH1A1KDM4C
SCHEMBL361255 0.84 KDM4E (0.58) NPSR1L3MBTL1KDM4EALDH1A1KDM4C
SCHEMBL31027302 0.84 KDM4E (0.58) NPSR1L3MBTL1KDM4EALDH1A1KDM4C
SCHEMBL277948 0.83 PDE3B (0.45) NPSR1L3MBTL1KDM4EALDH1A1TSHR
SCHEMBL871602 0.80 NPSR1 (0.50) NPSR1L3MBTL1KDM4EALDH1A1KDM4C
SCHEMBL162243 0.80 L3MBTL1 (0.53) NPSR1L3MBTL1KDM4EALDH1A1KDM4C
SCHEMBL29409978 0.80 NPSR1 (0.50) NPSR1L3MBTL1KDM4EALDH1A1KDM4C
SCHEMBL360639 0.80 NPSR1 (0.50) NPSR1L3MBTL1KDM4EALDH1A1KDM4C
SCHEMBL261104 0.78 NPSR1 (0.48) NPSR1L3MBTL1KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016101119-A1 FUSED HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-06-30 WO disclosed
US-5098462-A Herbicides SANDOZ LTD. (CH) 1992-03-24 US disclosed
US-5098466-A Herbicides SANDOZ LTD. (CH) 1992-03-24 US disclosed