SCHEMBL261104

SCHEMBL261104

COC(=O)c1nccnc1N

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.48
PRKCI P41743 6/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
ATR Q13535 1/20 0.47
NPC1 O15118 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
GRM5 P41594 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GBA1 P04062 1/20 0.44
TLR7 Q9NYK1 1/20 0.44
MLKL Q8NB16 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32682741 1.00 NPSR1 (0.48) NPSR1PRKCIL3MBTL1ATRNPC1
Hydrochloric Acid SCHEMBL5773639 0.98 NPSR1 (0.46) NPSR1PRKCIL3MBTL1ATRNPC1
SCHEMBL71518 0.84 NPSR1 (0.59) NPSR1L3MBTL1TDP1KDM4EALDH1A1
Dimethylamine SCHEMBL4391998 0.81 GBA1 (0.43) PRKCIL3MBTL1ATRNPC1TDP1
SCHEMBL2484699 0.79 GBA1 (0.44) PRKCIL3MBTL1ATRNPC1TDP1
SCHEMBL29642902 0.79 RAB9A (0.55) L3MBTL1NPC1TDP1KDM4EALDH1A1
SCHEMBL3979132 0.79 RAB9A (0.55) L3MBTL1NPC1TDP1KDM4EALDH1A1
SCHEMBL9632764 0.78 NPSR1 (0.52) NPSR1L3MBTL1KDM4EALDH1A1GAA
SCHEMBL8934162 0.78 NPC1 (0.39) PRKCIL3MBTL1ATRNPC1TDP1
SCHEMBL361255 0.77 KDM4E (0.58) NPSR1L3MBTL1KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 893 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119264345-A Porous adsorption resin for purifying silane and preparation method thereof 成都至诚大公光电科技有限公司 2025-01-07 CN claimed
CN-117946013-B Method for synthesizing 5, 6-dihalogen-3-aminopyrazine-2-methyl formate by one-pot method 白银康寓信生物科技有限公司 2024-07-02 CN claimed
CN-117946013-A Method for synthesizing 5, 6-dihalogen-3-aminopyrazine-2-methyl formate by one-pot method 白银康寓信生物科技有限公司 2024-04-30 CN claimed
CN-105327609-A Treating agent for removing three kinds of dioxin-like compounds in waste incineration waste off gas CHEN YIJUN 2016-02-17 CN claimed
CN-105327598-A Treating method for removing three kinds of dioxin-like compounds in waste incineration waste off gas CHEN YIJUN 2016-02-17 CN claimed
CN-105037281-A Preparation method for 3-(3-fluorophenoxyl)pyrazine-2-carboxylic acid CHANGSHA SHENCHENG BIOLOG SCIENCE & TECHNOLOGY CO LTD 2015-11-11 CN claimed
CN-105017166-A Preparation method of 3-(3-bromine phenoxy) pyrazine-2-carboxylic acid CHANGSHA SHENCHENG BIOLOG TECHNOLOGY CO LTD 2015-11-04 CN claimed
CN-104961691-A Preparation method of 3-(2-fluorophenoxy) pyrazine-2-carboxylic acid CHANGSHA SHENCHENG BIOTECHNOLOGY CO LTD 2015-10-07 CN claimed
CN-104961690-A Preparation method of 3-(4-fluorophenoxy) pyrazine-2-carboxylic acid CHANGSHA SHENCHENG BIOTECHNOLOGY CO LTD 2015-10-07 CN claimed
CN-102775358-A Preparation method of 6-fluoro-3-hydroxy-2-pyrazinamide SHANDONG QIDU PHARMACEUTICAL 2012-11-14 CN claimed
JP-3066675-A None JP disclosed
CN-115215923-B Macrocyclic broad-spectrum antibiotics 豪夫迈·罗氏有限公司 2026-05-19 CN disclosed
CN-115835909-B Cannabinoid receptor type 2 (CB 2) modulators and uses thereof 泰昂治疗公司 2026-05-15 CN disclosed
US-20250270202-A1 SUBSTITUTED 4-AMINOISOINDOLINE COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2025-08-28 US disclosed
EP-4373817-B1 SUBSTITUTED PYRAZINE-2-CARBOXAMIDES AS HPK1 INHIBITORS FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2025-05-21 EP disclosed
US-RE30563-E Preparation of benzoylureas ELI LILLY AND COMPANY (US) 1981-03-31 US disclosed
US-4160834-A INSECTICIDES ELI LILLY AND COMPANY (US) 1979-07-10 US disclosed
US-4133956-A Preparation of benzoylureas ELI LILLY AND COMPANY (US) 1979-01-09 US disclosed
US-4083977-A Novel insecticidal 1-(substituted benzoyl)-3-(substituted pyrazinyl)ureas ELI LILLY AND COMPANY (US) 1978-04-11 US disclosed
US-3954753-A SEDATIVES, MUSCLE RELAXANTS, ANTICONVULSANTS HOFFMANN-LA ROCHE INC. (US) 1976-05-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250270202-A1 SUBSTITUTED 4-AMINOISOINDOLINE COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF CUL4B, CUL3, CUL4A NPSR1 2643/4885PRKCI 3588/4885L3MBTL1 3218/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.