SCHEMBL9633136

SCHEMBL9633136

FC(F)=C(F)CCSc1nnc(-c2nnc(-c3ccccc3)o2)o1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.55
SMN1; SMN2 Q16637 5/20 0.54
EGFR P00533 1/20 0.54
NPC1 O15118 5/20 0.53
RAB9A P51151 5/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C19 P33261 1/20 0.53
HPGD P15428 3/20 0.51
MAPK1 P28482 2/20 0.51
CASP3 P42574 1/20 0.51
SENP8 Q96LD8 1/20 0.51
SENP7 Q9BQF6 1/20 0.51
SENP6 Q9GZR1 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
GSK3B P49841 1/20 0.51
MAPT P10636 3/20 0.51
THRB P10828 2/20 0.51
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9632708 0.85 GLA (0.40) SMN1; SMN2NPC1RAB9AMAPK1GSK3B
SCHEMBL10364612 0.85 MAPT (0.56) SMN1; SMN2NPC1RAB9AHPGDMAPK1
SCHEMBL10364759 0.84 HTT (0.55) SMN1; SMN2NPC1RAB9AMAPK1MAPT
SCHEMBL10363894 0.84 MAPT (0.60) NPSR1SMN1; SMN2NPC1RAB9ACYP1A2
SCHEMBL10364618 0.82 MAPT (0.53) NPSR1SMN1; SMN2NPC1RAB9AGSK3B
SCHEMBL17068793 0.80 MAPT (0.74) NPSR1SMN1; SMN2EGFRNPC1RAB9A
SCHEMBL17068760 0.80 NPSR1 (0.60) NPSR1SMN1; SMN2EGFRNPC1RAB9A
SCHEMBL9633100 0.80 SMN1; SMN2 (0.41) NPSR1SMN1; SMN2EGFRNPC1RAB9A
SCHEMBL9631769 0.77 PKM (0.42) SMN1; SMN2NPC1RAB9AMAPTTHRB
SCHEMBL7025544 0.77 NPSR1 (0.56) NPSR1SMN1; SMN2EGFRNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5162349-A Mercaptobis/1,3,4-oxa- and -thiadiazoles/ CIBA-GEIGY CORPORATION (US) 1992-11-10 US claimed
EP-0364396-A1 Neumaticides and fungicides CIBA-GEIGY AG (CH) 1990-04-18 EP claimed
US-5162349-A Mercaptobis/1,3,4-oxa- and -thiadiazoles/ CIBA-GEIGY CORPORATION (US) 1992-11-10 US disclosed
EP-0364396-A1 Neumaticides and fungicides CIBA-GEIGY AG (CH) 1990-04-18 EP disclosed