SCHEMBL9633707

SCHEMBL9633707

COC(=O)c1ccc(Cc2cccc3ccc(CCCCC(=O)N(C)C)cc23)c(OC)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
NQO2 P16083 1/20 0.41
ATM Q13315 1/20 0.41
CYP4A11 Q02928 3/20 0.40
CYP4F2 P78329 2/20 0.40
MTNR1A P48039 10/20 0.40
MTNR1B P49286 3/20 0.40
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9633818 0.98 NQO2 (0.42) KMT2ANQO2ATMCYP4A11CYP4F2
SCHEMBL9634189 0.92 PLA2G4A (0.41) KMT2AATMMTNR1AMTNR1BCYP1A2
SCHEMBL9633121 0.90 PLA2G4A (0.42) KMT2AATMMTNR1AMTNR1BCYP1A2
SCHEMBL9634320 0.88 CYP1A2 (0.50) NQO2CYP4A11CYP4F2MTNR1AMTNR1B
SCHEMBL9634990 0.84
SCHEMBL9633779 0.83 CYSLTR2 (0.46)
SCHEMBL9633723 0.82
SCHEMBL9633677 0.80 P4HB (0.38) KMT2ANQO2ATMMTNR1AALDH1A1
SCHEMBL9633679 0.80 P4HB (0.38) KMT2ANQO2ATMMTNR1AALDH1A1
SCHEMBL9633717 0.80 KMT2A (0.46) KMT2ANQO2MTNR1AMTNR1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337765-B1 ACYLSULFONAMIDE DERIVATIVES OF ALPHA-CARBOCYCLYLTOLUIC ACIDS USED AS LEUKOTRIENE ANTAGONISTS ICI AMERICAS INC. (US) 1992-10-14 EP disclosed
US-5095038-A Antiinflammatory, antiallergens ICI AMERICAS INC. (US) 1992-03-10 US disclosed
EP-0337765-A2 Acylsulfonamide derivatives of alpha-carbocyclyltoluic acids used as leukotriene antagonists ICI AMERICAS INC. (US) 1989-10-18 EP disclosed