SCHEMBL9634774

SCHEMBL9634774

COC(=O)C1C=CC(CC2=CCc3ccc(NC(=O)C(F)(F)F)cc32)(OC)C(OC)=C1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 6/20 0.41
MTNR1A P48039 6/20 0.41
MTNR1B P49286 6/20 0.41
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPY5R Q15761 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.31
MAPT P10636 1/20 0.31
KDM4E B2RXH2 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9634778 0.72 NQO2 (0.40) NQO2MTNR1AMTNR1BCYP1A2CYP2C9
SCHEMBL9635012 0.66 CYP1A2 (0.46) NQO2MTNR1AMTNR1BCYP1A2CYP2C9
SCHEMBL9634711 0.66 NQO2 (0.41) NQO2MTNR1AMTNR1BCYP1A2CYP2C9
SCHEMBL7785010 0.59 MTNR1A (1.00) NQO2MTNR1AMTNR1B
SCHEMBL4440336 0.57 CYP1A2 (1.00) CYP1A2CYP2C9CYP2C19L3MBTL1MAPT
SCHEMBL9633688 0.56 BAZ1A (0.51) CYP1A2CYP2C9CYP2C19NPY5RL3MBTL1
SCHEMBL14720795 0.56 CYP1A2 (0.75) CYP1A2CYP2C9CYP2C19NPY5RL3MBTL1
SCHEMBL8424252 0.56 CYP1A2 (0.60) CYP1A2CYP2C9CYP2C19L3MBTL1
SCHEMBL6422179 0.55 CYP1A2 (0.73) CYP1A2CYP2C9CYP2C19NPY5RL3MBTL1
SCHEMBL23088434 0.55 CYP1A2 (0.77) CYP1A2CYP2C9CYP2C19L3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337765-B1 ACYLSULFONAMIDE DERIVATIVES OF ALPHA-CARBOCYCLYLTOLUIC ACIDS USED AS LEUKOTRIENE ANTAGONISTS ICI AMERICAS INC. (US) 1992-10-14 EP disclosed
US-5095038-A Antiinflammatory, antiallergens ICI AMERICAS INC. (US) 1992-03-10 US disclosed
EP-0337765-A2 Acylsulfonamide derivatives of alpha-carbocyclyltoluic acids used as leukotriene antagonists ICI AMERICAS INC. (US) 1989-10-18 EP disclosed