SCHEMBL9636409

SCHEMBL9636409

NC1C=Cc2ccccc2OC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.36
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.33
CA2 P00918 1/20 0.33
ITGB2 P05107 1/20 0.33
ICAM1 P05362 1/20 0.33
ITGAL P20701 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
DRD1 P21728 1/20 0.33
TBXA2R P21731 1/20 0.33
SLC6A2 P23975 1/20 0.33
ADRA1A P35348 1/20 0.33
DRD3 P35462 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11112282 0.74 CYP19A1 (0.40) NISCHKDM4EMEN1ALDH1A1MAPT
SCHEMBL7927161 0.74 ALOX5 (0.38) NISCHMEN1ALDH1A1KMT2AHTR1A
SCHEMBL10601545 0.73 RAB9A (0.33) NISCHALDH1A1ABCG2CA2ITGB2
Hydrochloric Acid SCHEMBL8120795 0.73 ALOX5 (0.38) NISCHMEN1ALDH1A1KMT2AHTR1A
Hydrochloric Acid SCHEMBL10603135 0.72 POLB (0.34) ALDH1A1CA2NPC1RAB9AL3MBTL1
SCHEMBL7927222 0.72 HTT (0.39) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL30821601 0.69 KDM4E (0.37) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL3069884 0.69 KDM4E (0.37) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL18365855 0.68 ABCG2 (0.50) NISCHABCG2CA2ITGB2ICAM1
SCHEMBL31412834 0.67 CHRNB4 (0.43) NISCHABCG2HTR1AADRA2ADRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0180889-B1 3-AMINO-2,3-DIHYDRO-1-BENZOXEPINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE COMPOUNDS Kali-Chemie Pharma GmbH (DE) 1989-06-07 EP claimed
US-4672062-A ANTIDEPRESSANTS KALI-CHEMIE PHARMA GMBH (DE) 1987-06-09 US claimed
US-5084007-A Method for chemical promotion of the effects of low current transcranial electrostimulation MALIN DAVID H (US) 1992-01-28 US disclosed
WO-1991001756-A1 METHOD FOR CHEMICAL PROMOTION OF THE EFFECTS OF LOW CURRENT TRANSCRANIAL ELECTROSTIMULATION SKOLNICK MALCOLM H (US) 1991-02-21 WO disclosed
EP-0180889-B1 3-AMINO-2,3-DIHYDRO-1-BENZOXEPINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE COMPOUNDS Kali-Chemie Pharma GmbH (DE) 1989-06-07 EP disclosed
US-4672062-A ANTIDEPRESSANTS KALI-CHEMIE PHARMA GMBH (DE) 1987-06-09 US disclosed
US-4672062-A ANTIDEPRESSANTS KALI-CHEMIE PHARMA GMBH (DE) 1987-06-09 US disclosed
US-4672062-A ANTIDEPRESSANTS KALI-CHEMIE PHARMA GMBH (DE) 1987-06-09 US disclosed
EP-0180889-A2 3-Amino-2,3-dihydro-1-benzoxepine compounds, process for their preparation and medicaments containing these compounds Kali-Chemie Pharma GmbH (DE) 1986-05-14 EP disclosed