Piperazine

Piperazine

SCHEMBL964330

C1CNCCN1.C1CNCCN1.C=C

nearest known ligand 0.75

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ESR1

The experimentally established mechanism targets of Piperazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.75
MAPT P10636 1/20 0.75
PDE4A P27815 1/20 0.75
KDR P35968 1/20 0.75
CXCR4 P61073 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALDH1A1 P00352 1/20 0.42
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Piperazine SCHEMBL11729197 1.00 HIF1A (0.75) HIF1AMAPTPDE4AKDRCXCR4
Piperazine SCHEMBL2136219 1.00
Piperazine SCHEMBL5946680 0.94 HIF1A (0.67) HIF1AMAPTPDE4AKDRCXCR4
Piperazine SCHEMBL27797829 0.94
Aziridine SCHEMBL27781146 0.94
SCHEMBL576335 0.87 HIF1A (1.00) HIF1AMAPTPDE4AKDRCXCR4
Piperazine SCHEMBL734764 0.87 HIF1A (1.00) HIF1AMAPTPDE4AKDRCXCR4
SCHEMBL22003 0.87 HIF1A (1.00) HIF1AMAPTPDE4AKDRCXCR4
SCHEMBL3999265 0.87 HIF1A (1.00) HIF1AMAPTPDE4AKDRCXCR4
SCHEMBL577429 0.87 HIF1A (1.00) HIF1AMAPTPDE4AKDRCXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 129 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250320423-A1 METHOD FOR PREVENTING OR REDUCING LOW SPEED PRE-IGNITION IN DIRECT INJECTED SPARK-IGNITED ENGINES WITH MOLYBDENUM-CONTAINING LUBRICANT COMPOSITIONS CHEVRON ORONITE CO (US) 2025-10-16 US disclosed
EP-4608942-A2 METHOD FOR PREVENTING OR REDUCING LOW SPEED PRE-IGNITION IN DIRECT INJECTED SPARK-IGNITED ENGINES WITH MOLYBDENUM-CONTAINING LUBRICANT COMPOSITIONS Chevron Oronite Company LLC (US) 2025-09-03 EP disclosed
EP-4134414-B1 LUBRICATING OIL COMPOSITIONS CONTAINING ZIRCONIUM AND METHOD FOR PREVENTING OR REDUCING LOW SPEED PRE-IGNITION IN DIRECT INJECTED SPARK-IGNITED ENGINES CHEVRON USA INC (US) 2025-08-06 EP disclosed
EP-3652282-B1 LUBRICATING OIL COMPOSITIONS CONTAINING NON-SULFUR-PHOSPHORUS CONTAINING ZINC COMPOUNDS AND METHOD FOR PREVENTING OR REDUCING LOW SPEED PRE-IGNITION IN DIRECT INJECTED SPARK-IGNITED ENGINES CHEVRON ORONITE CO (US) 2025-08-06 EP disclosed
US-20250188381-A1 LUBRICATING OIL COMPOSITIONS WITH IMPROVED OXIDATIVE PERFORMANCE COMPRISING ALKYLATED DIPHENYLAMINE ANTIOXIDANT AND CARBOXYLATE DETERGENTS CHEVRON ORONITE COMPANY LLC (US) 2025-06-12 US disclosed
EP-3802752-B1 METHOD FOR PREVENTING OR REDUCING LOW SPEED PRE-IGNITION IN DIRECT INJECTED SPARK-IGNITED ENGINES WITH MANGANESE-CONTAINING LUBRICANT CHEVRON USA INC (US) 2023-07-19 EP disclosed
US-20230085359-A1 LUBRICATING OIL COMPOSITIONS WITH IMPROVED OXIDATIVE PERFORMANCE COMPRISING ALKYLATED DIPHENYLAMINE ANTIOXIDANT AND SULFONATE DETERGENTS CHEVRON ORONITE COMPANY LLC (US) 2023-03-16 US disclosed
EP-4134414-A1 LUBRICATING OIL COMPOSITIONS CONTAINING ZIRCONIUM AND METHOD FOR PREVENTING OR REDUCING LOW SPEED PRE-IGNITION IN DIRECT INJECTED SPARK-IGNITED ENGINES Chevron U.S.A. Inc. (US) 2023-02-15 EP disclosed
EP-4118171-A1 LUBRICATING OIL COMPOSITIONS WITH IMPROVED OXIDATIVE PERFORMANCE COMPRISING ALKYLATED DIPHENYLAMINE ANTIOXIDANT AND SULFONATE DETERGENTS Chevron Oronite Company LLC (US) 2023-01-18 EP disclosed
EP-4118170-A1 LUBRICATING OIL COMPOSITIONS WITH IMPROVED OXIDATIVE PERFORMANCE COMPRISING ALKYLATED DIPHENYLAMINE ANTIOXIDANT AND CARBOXYLATE DETERGENTS Chevron Oronite Company LLC (US) 2023-01-18 EP disclosed
US-4369119-A Antioxidant combinations of molybdenum complexes and organic sulfur compounds for lubricating oils CHEVRON RESEARCH COMPANY (US) 1983-01-18 US disclosed
US-4285822-A OXIDATION RESISTANCE; OIL-SOLUBLE COMPLEX OF AN ACIDIC MOLYBDENUM COMPOUND, A BASIC NITROGEN-CONTAINING COMPOUND, AND CARBON DISULFIDE CHEVRON RESEARCH COMPANY (US) 1981-08-25 US disclosed
US-4283295-A BY REACTING AMMONIUM TETRATHIAMOLYBDATE AND A BASIC NITROGEN COMPOUND CHEVRON RESEARCH COMPANY (US) 1981-08-11 US disclosed
US-4272387-A Process of preparing molybdenum complexes, the complexes so-produced and lubricants containing same CHEVRON RESEARCH COMPANY (US) 1981-06-09 US disclosed
US-4265773-A Process of preparing molybdenum complexes, the complexes so-produced and lubricants containing same CHEVRON RESEARCH COMPANY (US) 1981-05-05 US disclosed
US-4263152-A OIL ADDITIVES COMPRISING A COMPLEX OF AN ACIDIC MOLYBDENUM COMPOUND, A BASIC NITROGEN-CONTAINING COMPOUND, AND A SULFUR SOURCE; OXIDATION RESISTANCE CHEVRON RESEARCH COMPANY (US) 1981-04-21 US disclosed
US-4261843-A Reaction product of acidic molybdenum compound with basic nitrogen compound and lubricants containing same CHEVRON RESEARCH COMPANY (US) 1981-04-14 US disclosed
US-4259194-A Reaction product of ammonium tetrathiomolybdate with basic nitrogen compounds and lubricants containing same CHEVRON RESEARCH COMPANY (US) 1981-03-31 US disclosed
US-4259195-A ANTIOXIDANT OIL ADDITIVES CHEVRON RESEARCH COMPANY (US) 1981-03-31 US disclosed
US-3951614-A REACTION PRODUCT OF A HYDROCARBYL AMINE AND POLYFUNCTIONAL COUPLING AGENT CHEVRON RESEARCH COMPANY (US) 1976-04-20 US disclosed