SCHEMBL9657223

SCHEMBL9657223

N#CC(C#N)=C(N)Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
LMNA P02545 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 2/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
AKR1B1 P15121 1/20 0.41
MAPT P10636 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HIF1A Q16665 1/20 0.39
GAA P10253 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP1B1 Q16678 1/20 0.38
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
IDO1 P14902 1/20 0.36
NOS3 P29474 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993215 0.79 CES1 (0.55) KMT2ALMNAMEN1CES2CES1
SCHEMBL3945284 0.78 KDM4E (0.45) KMT2ALMNAKDM4EMEN1CES2
SCHEMBL8967450 0.77 CES1 (0.43) KMT2ALMNAKDM4EMEN1CES2
SCHEMBL11765098 0.75 CES1 (0.41) KMT2ALMNAKDM4EMEN1CES2
SCHEMBL11010613 0.75 CES2 (0.41) KMT2AKDM4EMEN1CES2CES1
SCHEMBL12263802 0.75 CES1 (0.50) KMT2ALMNAMEN1CES2CES1
SCHEMBL4978892 0.74 CTSL (0.46) KMT2ALMNAMEN1CES2CES1
SCHEMBL955096 0.74 CES1 (0.56) KMT2ALMNAMEN1CES2CES1
SCHEMBL16550069 0.73 ALDH1A1 (0.43) KMT2AKDM4EMEN1CES2CES1
SCHEMBL21436188 0.71 NOS2 (0.48) KMT2ALMNAMEN1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0327981-B1 PROCESS FOR THE PREPARATION OF 2-CYANO-3-AMINOACRYL NITRILE DERIVATIVES BASF Aktiengesellschaft (DE) 1992-05-06 EP disclosed
US-5047570-A Reacting nitrile with alkanol inpresence of hydrogen halide, then with malodinitrile BASF AKTIENGESELLSCHAFT (DE) 1991-09-10 US disclosed
EP-0327981-A1 Process for the preparation of 2-cyano-3-aminoacryl nitrile derivatives BASF Aktiengesellschaft (DE) 1989-08-16 EP disclosed