SCHEMBL965845

SCHEMBL965845

CC1CN(c2c(F)cc3c(=O)c(C(=O)O)cn(C4CC4)c3c2Cl)CC(C)N1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.70
POLB P06746 3/20 0.70
OPRM1 P35372 2/20 0.70
CHRM2 P08172 1/20 0.70
CHRM1 P11229 1/20 0.70
OPRD1 P41143 1/20 0.70
MEN1 O00255 2/20 0.66
KMT2A Q03164 2/20 0.66
KCNH2 Q12809 6/20 0.62
KDM4E B2RXH2 5/20 0.62
HPGD P15428 5/20 0.62
HSD17B10 Q99714 4/20 0.62
PRKD3 O94806 1/20 0.62
ALOX15 P16050 1/20 0.62
CLK2 P49760 1/20 0.62
CLK4 Q9HAZ1 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
CACNA1F O60840 1/20 0.61
MAPK1 P28482 1/20 0.61
CACNA1D Q01668 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10695169 1.00 ALDH1A1 (0.70) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10586019 0.91 MEN1 (0.72) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9636636 0.91 MEN1 (0.72) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9522847 0.90 ALDH1A1 (0.72) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL8433684 0.90 ALDH1A1 (0.77) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL5792107 0.89 MEN1 (0.67) ALDH1A1POLBOPRM1CHRM2CHRM1
Hydrochloric Acid SCHEMBL10914782 0.89 ALDH1A1 (0.76) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9671640 0.88 ALDH1A1 (0.72) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10695174 0.88 ALDH1A1 (0.54) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10695974 0.88 ALDH1A1 (0.54) ALDH1A1POLBOPRM1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7867992-B2 such as 1-Cyclopropyl-N-(2,4-dichlorobenzyl)-6-fluoro-8-methoxy-7-[3-methyl-4-(2-{[(methylamino)carbonyl]amino}-2-oxoethyl)piperazin-1-yl]-4-oxo-1,4-dihydroquinoline-3-carboxamide, used for the treatment and/or prophylaxis of viral diseases or infections, particularly against cytomegaloviruses AICURIS GMBH & CO. KG (DE) 2011-01-11 US disclosed
US-7569563-B2 Substituted quinolones II AICURIS GMBH & CO. HK (DE) 2009-08-04 US disclosed
US-20080261964-A1 Substituted quinolones II AICURIS GMBH & CO. KG (DE) 2008-10-23 US disclosed
US-20070293478-A1 Substituted quinolones BAYER HEALTHCARE AG (DE) 2007-12-20 US disclosed
EP-1768973-B1 SUBSTITUTED QUINOLONES AICURIS GMBH & CO KG (DE) 2007-12-05 EP disclosed
EP-0178388-A1 Quinolinecarboxylic acid derivatives KYORIN PHARMACEUTICAL CO., LTD. (JP) 1986-04-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080261964-A1 Substituted quinolones II TOP2A, TPMT, TOP2B ALDH1A1 1587/4885POLB 37/4885OPRM1 3551/4885
US-20070293478-A1 Substituted quinolones IRF3, TPMT, NQO2 ALDH1A1 2853/4885POLB 86/4885OPRM1 3486/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.