SCHEMBL9668309

SCHEMBL9668309

CCOC(=O)CC(=O)CSCCNC=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.45
HSD17B10 Q99714 2/20 0.45
MGAM O43451 1/20 0.42
SI P14410 1/20 0.42
MGAM2 Q2M2H8 1/20 0.42
ADH1B P00325 3/20 0.38
ADH1A P07327 3/20 0.38
ADH7 P40394 3/20 0.38
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
ADH1C P00326 2/20 0.36
EPHX1 P07099 1/20 0.35
ADH4 P08319 1/20 0.35
ALDH1A1 P00352 5/20 0.34
HTT P42858 3/20 0.34
MAPK1 P28482 2/20 0.34
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9668780 0.84 FAAH (0.32) GAAHSD17B10ADH1BADH1AADH7
SCHEMBL10959041 0.81 GAA (0.54) GAAHSD17B10MGAMSIMGAM2
SCHEMBL9824473 0.78 GAA (0.50) GAAHSD17B10MGAMSIMGAM2
SCHEMBL11451516 0.78 HSD17B10 (0.50) GAAHSD17B10MGAMSIMGAM2
SCHEMBL9668772 0.77 FAAH (0.31) ADH1BADH1AADH7
SCHEMBL10517462 0.76 ADH1B (0.37) HSD17B10ADH1BADH1AADH7ADH1C
SCHEMBL3388745 0.76 GAA (0.56) GAAHSD17B10MGAMSIMGAM2
SCHEMBL8866115 0.76 CES2 (0.55) GAAHSD17B10MGAMSIMGAM2
SCHEMBL9667017 0.75 NPSR1 (0.40) ADH1BADH1AADH7ADH1CMAPT
SCHEMBL9667011 0.75 NPSR1 (0.40) ADH1BADH1AADH7ADH1CMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0312541-B1 2-(AMINOALKYLTHIO)METHYL-1,4-DIHYDROPYRIDINE, A METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-08-26 EP disclosed
EP-0254064-B1 2-(AMINOALKYLTHIO)METHYL-1,4-DIHYDROPYRIDINE, A METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-06-17 EP disclosed
US-5047414-A Hypotensive agents BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1991-09-10 US disclosed
EP-0312541-A1 2-(AMINOALKYLTHIO)METHYL-1,4-DIHYDROPYRIDINE, A METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. BOEHRINGER BIOCHEMIA SRL (IT) 1989-04-26 EP disclosed
EP-0254064-A1 2-(Aminoalkylthio)methyl-1,4-dihydropyridine, a method for the preparation thereof and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1988-01-27 EP disclosed
WO-1988000187-A1 2-(AMINOALKYLTHIO)METHYL-1,4-DIHYDROPYRIDINE, A METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1988-01-14 WO disclosed