SCHEMBL9668538

SCHEMBL9668538

Cc1ccc(N(C(=O)[C@@H](N)Cc2cnc[nH]2)c2ccccc2N)cc1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NLN Q9BYT8 4/20 0.48
CYP3A4 P08684 1/20 0.46
SLC7A5 Q01650 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Histidine SCHEMBL27702202 0.75 CYP3A4 (0.78) NLNCYP3A4SLC7A5
SCHEMBL18809892 0.71 CYP3A4 (0.67) NLNCYP3A4SLC7A5
Histidine SCHEMBL27676546 0.70 CYP3A4 (0.78) NLNCYP3A4SLC7A5
SCHEMBL6037588 0.69 TRPM8 (0.40)
SCHEMBL5702193 0.69 CYP3A4 (0.55) CYP3A4SLC7A5
SCHEMBL3632930 0.67 CYP3A4 (0.60) NLNCYP3A4SLC7A5
SCHEMBL18162806 0.67 CYP3A4 (0.73) CYP3A4SLC7A5
SCHEMBL13609239 0.67 CYP3A4 (0.73) CYP3A4SLC7A5
SCHEMBL7962292 0.67 CYP3A4 (0.73) CYP3A4SLC7A5
Histidine SCHEMBL27388700 0.66 CYP3A4 (0.88) NLNCYP3A4SLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0485458-A1 THIOACYLATING REAGENTS AND INTERMEDIATES, THIOPEPTIDES, AND METHODS FOR PREPARING AND USING SAME. IAF BIOCHEM INT (CA) 1992-05-20 EP claimed
WO-1991001976-A1 THIOACYLATING REAGENTS AND INTERMEDIATES, THIOPEPTIDES, AND METHODS FOR PREPARING AND USING SAME IAF BIOCHEM INTERNATIONAL INC. (CA) 1991-02-21 WO claimed