SCHEMBL9669331

SCHEMBL9669331

Nc1cccc2ccc3nc(O)c(O)nc3c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.45
PLAU P00749 2/20 0.39
NCF1 P14598 1/20 0.39
MET P08581 1/20 0.38
JAK2 O60674 1/20 0.37
RPS6KA3 P51812 1/20 0.37
MELK Q14680 1/20 0.37
STK24 Q9Y6E0 1/20 0.37
ACHE P22303 1/20 0.36
ALDH1A1 P00352 5/20 0.36
HPGD P15428 4/20 0.36
HSD17B10 Q99714 3/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 2/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1B1 Q16678 1/20 0.36
KMT2A Q03164 3/20 0.34
KDM4E B2RXH2 3/20 0.34
GAA P10253 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2865383 0.80 ACHE (0.46) PLAUNCF1ACHEALDH1A1HPGD
SCHEMBL9669419 0.76 SOS2 (0.39) PLAUACHEALDH1A1HPGDHSD17B10
SCHEMBL9670587 0.74 TYMS (0.49) TYMSALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL9534423 0.72 MAPT (0.39) ACHECYP1A2KMT2AKDM4EGAA
SCHEMBL10085320 0.72 ACHE (0.58) PLAUNCF1ACHEALDH1A1HPGD
SCHEMBL14742902 0.72 ALDH1A1 (0.59) TYMSPLAUMETJAK2RPS6KA3
Hydrochloric Acid SCHEMBL11047993 0.71 MAPT (0.38) ACHECYP1A2KMT2AKDM4EGAA
SCHEMBL9578558 0.71 PRMT5 (0.49) ALDH1A1HSD17B10CYP1A2CYP3A4TSHR
SCHEMBL65699 0.70 JAK2 (0.54) TYMSJAK2RPS6KA3MELKSTK24
SCHEMBL29349435 0.70 JAK2 (0.54) TYMSJAK2RPS6KA3MELKSTK24

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4889855-A ADMINISTERING GLUTAMATE ANTAGONIST TO INHIBIT HYPERACTIVITY OF EXCITATORY NEUROTRANSMITTERS A/S FERROSAN (DK) 1989-12-26 US claimed
EP-0283959-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-01-02 EP disclosed
US-4912108-A Containing hydroxy substitution A/S FERROSAN (DK) 1990-03-27 US disclosed
US-4889855-A ADMINISTERING GLUTAMATE ANTAGONIST TO INHIBIT HYPERACTIVITY OF EXCITATORY NEUROTRANSMITTERS A/S FERROSAN (DK) 1989-12-26 US disclosed
EP-0283959-A1 Heterocyclic compounds and their preparation and use NOVO NORDISK A/S (DK) 1988-09-28 EP disclosed