SCHEMBL9670587

SCHEMBL9670587

O=[N+]([O-])c1cccc2ccc3nc(O)c(O)nc3c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.49
GPR35 Q9HC97 2/20 0.44
PDE10A Q9Y233 1/20 0.44
NOS1 P29475 2/20 0.43
NOS2 P35228 2/20 0.43
CYP1A2 P05177 3/20 0.43
ALDH1A1 P00352 3/20 0.43
HSP90AA1 P07900 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C19 P33261 2/20 0.43
TP53 P04637 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX15 P16050 1/20 0.43
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
HSP90AB1 P08238 1/20 0.42
MAPT P10636 2/20 0.41
HTT P42858 1/20 0.41
ERN1 O75460 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2863690 0.82 MEN1 (0.59) GPR35PDE10ANOS1NOS2CYP1A2
SCHEMBL9669275 0.79 ALDH1A1 (0.44) GPR35CYP1A2ALDH1A1HSP90AA1CYP2C19
SCHEMBL9670143 0.77 KDM4E (0.52) GPR35PDE10ANOS1NOS2CYP1A2
SCHEMBL9670624 0.76 EGFR (0.42) GPR35PDE10ANOS1NOS2CYP1A2
SCHEMBL28610797 0.74 GPR35 (0.44) GPR35ALDH1A1HSP90AA1CYP3A4TP53
SCHEMBL29626558 0.74 ALDH1A1 (0.61) TYMSGPR35PDE10ANOS1NOS2
SCHEMBL187697 0.74 ALDH1A1 (0.61) TYMSGPR35PDE10ANOS1NOS2
SCHEMBL9669331 0.74 TYMS (0.45) TYMSCYP1A2ALDH1A1CYP3A4CYP2C19
SCHEMBL2927810 0.73 GPR35 (0.60) TYMSGPR35PDE10ANOS1NOS2
SCHEMBL18416514 0.73 PDE10A (0.75) PDE10ACYP1A2ALDH1A1HSP90AA1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0283959-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-01-02 EP disclosed
US-4912108-A Containing hydroxy substitution A/S FERROSAN (DK) 1990-03-27 US disclosed
US-4889855-A ADMINISTERING GLUTAMATE ANTAGONIST TO INHIBIT HYPERACTIVITY OF EXCITATORY NEUROTRANSMITTERS A/S FERROSAN (DK) 1989-12-26 US disclosed
EP-0283959-A1 Heterocyclic compounds and their preparation and use NOVO NORDISK A/S (DK) 1988-09-28 EP disclosed