SCHEMBL9669809

SCHEMBL9669809

Nc1c([N+](=O)[O-])ccc2c(Br)cccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSB P07858 2/20 0.58
TDP1 Q9NUW8 4/20 0.47
ALDH1A1 P00352 7/20 0.43
CYP3A4 P08684 3/20 0.43
MAPT P10636 4/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALOX15 P16050 2/20 0.41
TSHR P16473 2/20 0.41
KDM4E B2RXH2 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP1A2 P05177 1/20 0.41
MAPK1 P28482 1/20 0.41
NOS1 P29475 1/20 0.41
CYP2C19 P33261 1/20 0.41
NOS2 P35228 1/20 0.41
BLM P54132 1/20 0.41
HSD17B10 Q99714 1/20 0.40
GAA P10253 1/20 0.38
TTR P02766 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30881743 1.00 CTSB (0.58) CTSBTDP1ALDH1A1CYP3A4MAPT
SCHEMBL16204105 0.83 TDP1 (0.50) CTSBTDP1ALDH1A1CYP3A4MAPT
SCHEMBL9363144 0.82 CTSB (0.77) CTSBTDP1ALDH1A1CYP3A4MAPT
SCHEMBL30064818 0.82 CTSB (0.77) CTSBTDP1ALDH1A1CYP3A4MAPT
SCHEMBL2963038 0.80 TDP1 (0.75) CTSBTDP1ALDH1A1CYP3A4MAPT
SCHEMBL2255970 0.80 ALDH1A1 (0.55) CTSBTDP1ALDH1A1CYP3A4MAPT
SCHEMBL29643206 0.80 TDP1 (0.75) CTSBTDP1ALDH1A1CYP3A4MAPT
SCHEMBL8722948 0.76 TDP1 (0.61) CTSBTDP1ALDH1A1CYP3A4MAPT
SCHEMBL9669943 0.76 CTSB (0.43) CTSBTDP1ALDH1A1CYP3A4MAPT
SCHEMBL8687725 0.74 CTSB (0.77) CTSBTDP1ALDH1A1CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0283959-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-01-02 EP disclosed
US-4912108-A Containing hydroxy substitution A/S FERROSAN (DK) 1990-03-27 US disclosed
US-4889855-A ADMINISTERING GLUTAMATE ANTAGONIST TO INHIBIT HYPERACTIVITY OF EXCITATORY NEUROTRANSMITTERS A/S FERROSAN (DK) 1989-12-26 US disclosed
EP-0283959-A1 Heterocyclic compounds and their preparation and use NOVO NORDISK A/S (DK) 1988-09-28 EP disclosed