SCHEMBL9680321

SCHEMBL9680321

CCc1cc(NCc2cc3c(nc2OC)CCCC3)c(=O)[nH]c1CO

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KDM4E B2RXH2 5/20 0.32
MAPT P10636 6/20 0.31
POLB P06746 2/20 0.31
GAA P10253 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HIF1A Q16665 1/20 0.31
APAF1 O14727 1/20 0.31
RECQL P46063 1/20 0.31
TP53 P04637 2/20 0.30
THRB P10828 1/20 0.30
P2RX7 Q99572 1/20 0.30
NPC1 O15118 1/20 0.30
NFKB1 P19838 1/20 0.30
RAB9A P51151 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681437 0.98 NPSR1 (0.34) NPSR1RXFP1KDM4EMAPTGAA
SCHEMBL9846089 0.87 NPSR1 (0.38) NPSR1RXFP1KDM4EMAPTPOLB
SCHEMBL9682084 0.86 MAPT (0.36) NPSR1RXFP1KDM4EMAPTPOLB
SCHEMBL9681383 0.84 NPC1 (0.34) NPSR1RXFP1KDM4EMAPTPOLB
SCHEMBL9846123 0.82 NPSR1 (0.36) NPSR1RXFP1KDM4EMAPTPOLB
SCHEMBL9681299 0.81 MAPT (0.35) KDM4EMAPTPOLBGAAALDH1A1
SCHEMBL9681421 0.81 MAPT (0.37) KDM4EMAPTPOLBGAAALDH1A1
SCHEMBL9680861 0.81 SLC2A1 (0.38) KDM4EMAPTPOLBGAAALDH1A1
SCHEMBL9681349 0.78 MAPT (0.40) KDM4EMAPTGAAALDH1A1HIF1A
SCHEMBL9846183 0.73 RXFP1 (0.38) NPSR1RXFP1KDM4EMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP claimed
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed