SCHEMBL9846183

SCHEMBL9846183

CCc1cc(NCc2nc3c(cc2OC)CCCC3)c(=O)[nH]c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPT P10636 3/20 0.36
POLB P06746 2/20 0.36
KDM4E B2RXH2 2/20 0.35
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
NPC1 O15118 2/20 0.34
TP53 P04637 2/20 0.33
THRB P10828 1/20 0.33
ALDH1A1 P00352 4/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
P2RX7 Q99572 1/20 0.33
PPARG P37231 1/20 0.33
KMT2A Q03164 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
SLC2A1 P11166 1/20 0.33
GAA P10253 1/20 0.32
HIF1A Q16665 1/20 0.32
APAF1 O14727 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9682084 0.87 MAPT (0.36) RXFP1NPSR1MAPTPOLBKDM4E
SCHEMBL9846089 0.85 NPSR1 (0.38) RXFP1NPSR1MAPTPOLBKDM4E
SCHEMBL9681383 0.85 NPC1 (0.34) RXFP1NPSR1MAPTPOLBKDM4E
SCHEMBL9846212 0.81 SLC2A1 (0.40) MAPTPOLBKDM4EPDE3BPDE3A
SCHEMBL9846203 0.81 PDE3B (0.38) MAPTKDM4EPDE3BPDE3AALDH1A1
SCHEMBL9846298 0.81 PDE3B (0.38) MAPTKDM4EPDE3BPDE3ASMN1; SMN2
SCHEMBL9846175 0.79 PDE3B (0.38) MAPTPOLBKDM4EPDE3BPDE3A
SCHEMBL9846123 0.76 NPSR1 (0.36) RXFP1NPSR1MAPTPOLBKDM4E
SCHEMBL27337641 0.73 POLB (0.49) MAPTPOLBKDM4EPDE3BPDE3A
SCHEMBL9680321 0.73 NPSR1 (0.36) RXFP1NPSR1MAPTPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed