SCHEMBL9680865

SCHEMBL9680865

CC(=O)c1cc(NCc2nc3c(Cl)ccc(Cl)c3o2)c(=O)[nH]c1C

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
CD38 P28907 12/20 0.32
CYP3A4 P08684 4/20 0.32
KCNH2 Q12809 1/20 0.32
BRD4 O60885 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
L-697661 SCHEMBL599639 0.84 FABP4 (0.34) NPC1
SCHEMBL9283257 0.83 ADRA2A (0.32)
SCHEMBL9456135 0.83
SCHEMBL9846262 0.82 IDH1 (0.34) GAAPDE3BPDE3A
SCHEMBL9455992 0.78 HCAR2 (0.33)
SCHEMBL9171193 0.77 FABP4 (0.34) CD38CYP3A4
SCHEMBL9846309 0.76 FABP4 (0.31) NPC1
SCHEMBL9846072 0.76 TYMS (0.32)
SCHEMBL9680329 0.73 PTGES (0.31)
SCHEMBL9846215 0.73 FABP4 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP claimed
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed