SCHEMBL9455992

SCHEMBL9455992

CCc1cc(NCc2nc3c(Cl)ccc(Cl)c3o2)c(=O)[nH]c1CO

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.33
FABP4 P15090 1/20 0.32
IDH1 O75874 4/20 0.31
TYMS P04818 1/20 0.31
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846309 0.92 FABP4 (0.31) HCAR2FABP4MEN1ALDH1A1HPGD
SCHEMBL9846072 0.90 TYMS (0.32) FABP4IDH1TYMSMEN1ALDH1A1
L-697661 SCHEMBL599639 0.86 FABP4 (0.34) FABP4IDH1TYMSMEN1ALDH1A1
L-697661 SCHEMBL29456987 0.86 FABP4 (0.34) FABP4IDH1TYMSMEN1ALDH1A1
SCHEMBL9681878 0.84 KMT2A (0.35) HCAR2MEN1ALDH1A1HPGDKMT2A
SCHEMBL9680329 0.83 PTGES (0.31)
SCHEMBL9601892 0.82 ALDH1A1 (0.36) HCAR2TYMSMEN1ALDH1A1HPGD
SCHEMBL9171193 0.79 FABP4 (0.34) FABP4IDH1TYMS
SCHEMBL9680865 0.78 NPC1 (0.33)
SCHEMBL9846215 0.77 FABP4 (0.31) FABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP claimed
US-5200329-A An Isolating Compound Which is Useful in the Prevention or Tre atment of HIV Infection and the Treatment of AIDS MERCK & CO., INC. (US) 1993-04-06 US disclosed
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed