SCHEMBL9680995

SCHEMBL9680995

NNC(=O)c1[c]ccc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 2/20 0.38
GFER P55789 2/20 0.34
MPO P05164 2/20 0.34
CYP3A4 P08684 2/20 0.34
BLM P54132 2/20 0.34
KDM5A P29375 1/20 0.34
PMP22 Q01453 1/20 0.34
HIF1A Q16665 1/20 0.34
ALDH1A1 P00352 7/20 0.34
KDM4E B2RXH2 5/20 0.34
HDAC1 Q13547 2/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MAPT P10636 4/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
LMNA P02545 2/20 0.33
NSD2 O96028 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3991217 0.81 GAA (0.39) ALDH1A1KDM4EHDAC1CA2HDAC6
SCHEMBL7212212 0.80 PARP1 (0.45) CYP3A4ALDH1A1CYP1A2CYP2C19
SCHEMBL10636542 0.78 KDM4E (0.37) ALPLGFERMPOCYP3A4BLM
SCHEMBL6204339 0.78 ALDH1A1 (0.49) ALPLGFERMPOCYP3A4BLM
SCHEMBL5759254 0.77 ALDH1A1 (0.43) CYP3A4ALDH1A1KDM4EMAPTL3MBTL1
SCHEMBL4321490 0.76 KEAP1 (0.39) HIF1AALDH1A1KDM4ECA1CA2
SCHEMBL27707510 0.75 CES2 (0.33) ALDH1A1
SCHEMBL27952340 0.74 TRPM8 (0.35) CYP3A4ALDH1A1MAPTL3MBTL1GAA
SCHEMBL3982238 0.74 MEN1 (0.42) ALPLALDH1A1KDM4EMAPTL3MBTL1
SCHEMBL4147070 0.73 NPC1 (0.57) HDAC1CA2HDAC6POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed