SCHEMBL9681007

SCHEMBL9681007

CC(=Cc1ccccc1C=O)C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 1/20 0.42
THRB P10828 1/20 0.42
BLM P54132 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ERN1 O75460 3/20 0.37
TLR2 O60603 1/20 0.37
TLR1 Q15399 1/20 0.37
TLR6 Q9Y2C9 1/20 0.37
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
TRIM24 O15164 1/20 0.36
TRIM33 Q9UPN9 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
HTT P42858 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ELANE P08246 1/20 0.33
PRTN3 P24158 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680999 1.00 MEN1 (0.42) MEN1KMT2ALMNATHRBBLM
SCHEMBL31065882 0.85 ERN1 (0.39) ERN1TLR2TLR1TLR6TRIM24
SCHEMBL9681561 0.80 MEN1 (0.38) MEN1KMT2ALMNATHRBBLM
SCHEMBL9681557 0.80 MEN1 (0.38) MEN1KMT2ALMNATHRBBLM
SCHEMBL28915528 0.78 AKR1C3 (0.58) MEN1KMT2ATDP1ALDH1A1TSHR
SCHEMBL20853874 0.78 AKR1C3 (0.58) MEN1KMT2ATDP1ALDH1A1TSHR
SCHEMBL7009992 0.78 ALDH1A1 (0.39) MEN1KMT2ALMNAALDH1A1BCHE
SCHEMBL7009987 0.78 ALDH1A1 (0.39) MEN1KMT2ALMNAALDH1A1BCHE
SCHEMBL9680987 0.77 KMT2A (0.50) MEN1KMT2ALMNATHRBBLM
SCHEMBL9680982 0.77 KMT2A (0.50) MEN1KMT2ALMNATHRBBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5162345-A Dihydropyridinedicarboxylate Derivatives GLAXO, S.P.A. (IT) 1992-11-10 US disclosed
US-5091395-A Hypotensive agents GLAXO S.P.A. (IT) 1992-02-25 US disclosed
EP-0226271-B1 1,4-DIHYDROPYRIDINE COMPOUNDS AND THEIR PREPARATION AND PHARMACEUTICAL FORMULATION GLAXO S.p.A. (IT) 1990-11-22 EP disclosed
EP-0226271-A1 1,4-Dihydropyridine compounds and their preparation and pharmaceutical formulation GLAXO S.p.A. (IT) 1987-06-24 EP disclosed