SCHEMBL9681561

SCHEMBL9681561

CCC(=Cc1ccccc1C=O)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.38
LMNA P02545 3/20 0.38
KMT2A Q03164 3/20 0.38
THRB P10828 1/20 0.38
BLM P54132 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.36
PLIN1 O60240 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
PLIN5 Q00G26 1/20 0.35
ABHD5 Q8WTS1 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HTT P42858 2/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP2C19 P33261 3/20 0.33
TSHR P16473 1/20 0.33
TRIM24 O15164 1/20 0.33
TRIM33 Q9UPN9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681557 1.00 MEN1 (0.38) MEN1LMNAKMT2ATHRBBLM
SCHEMBL9681733 0.82 MAPT (0.49) MEN1LMNAKMT2ATHRBBLM
SCHEMBL9681724 0.82 MAPT (0.49) MEN1LMNAKMT2ATHRBBLM
SCHEMBL9680999 0.80 MEN1 (0.42) MEN1LMNAKMT2ATHRBBLM
SCHEMBL9681007 0.80 MEN1 (0.42) MEN1LMNAKMT2ATHRBBLM
SCHEMBL9737066 0.79 ALDH1A1 (0.38) MEN1LMNAKMT2AMAPTALDH1A1
SCHEMBL5606940 0.73 MIF (0.46) MEN1LMNAKMT2AMAPTALDH1A1
SCHEMBL9680642 0.71 MAPT (0.47) MEN1LMNAKMT2ATHRBBLM
SCHEMBL29262005 0.70 MEN1 (0.36) MEN1LMNAKMT2ATHRBBLM
SCHEMBL28562985 0.70 HSD11B1 (0.41) MEN1LMNAKMT2APLIN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5162345-A Dihydropyridinedicarboxylate Derivatives GLAXO, S.P.A. (IT) 1992-11-10 US disclosed
US-5091395-A Hypotensive agents GLAXO S.P.A. (IT) 1992-02-25 US disclosed
EP-0226271-B1 1,4-DIHYDROPYRIDINE COMPOUNDS AND THEIR PREPARATION AND PHARMACEUTICAL FORMULATION GLAXO S.p.A. (IT) 1990-11-22 EP disclosed
EP-0226271-A1 1,4-Dihydropyridine compounds and their preparation and pharmaceutical formulation GLAXO S.p.A. (IT) 1987-06-24 EP disclosed