SCHEMBL9681353

SCHEMBL9681353

CP(C)(=O)CN1CCN(c2nn(-c3ccccc3)c3ccccc23)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 5/20 0.42
PTGER1 P34995 2/20 0.42
ALDH1A1 P00352 5/20 0.41
KMT2A Q03164 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.40
GFER P55789 1/20 0.40
KDM4E B2RXH2 2/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 4/20 0.38
MAPT P10636 3/20 0.38
GLA P06280 1/20 0.38
DRD3 P35462 1/20 0.38
MEN1 O00255 2/20 0.37
HTT P42858 1/20 0.37
POLB P06746 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680605 0.81 DRD2 (0.57) KHKALDH1A1KDM4ENPC1LMNA
SCHEMBL9682450 0.81 DRD4 (0.58) KHKALDH1A1KDM4ELMNAMAPT
SCHEMBL9680621 0.80 KHK (0.44) KHKPTGER1ALDH1A1KMT2ACYP1A2
SCHEMBL9680636 0.80 SMO (0.50) KHKPTGER1ALDH1A1KMT2ATSHR
SCHEMBL6125292 0.79 KHK (0.56) KHKPTGER1ALDH1A1KDM4E
SCHEMBL9681250 0.79 HTR1A (0.60) ALDH1A1LMNAMAPTPOLBMAPK1
SCHEMBL9681419 0.79 KDM4E (0.49) PTGER1ALDH1A1KMT2ATSHRKDM4E
SCHEMBL9680805 0.78 DRD3 (0.43) KHKPTGER1ALDH1A1KDM4ENPC1
Hydrochloric Acid SCHEMBL9682152 0.78 KHK (0.54) KHKPTGER1ALDH1A1KDM4E
SCHEMBL9682466 0.78 DRD3 (0.47) KHKPTGER1ALDH1A1CYP2D6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed