SCHEMBL9681250

SCHEMBL9681250

c1ccc(CCN2CCN(c3nn(-c4ccccc4)c4ccccc34)CC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.60
DRD2 P14416 1/20 0.60
MAPT P10636 3/20 0.58
ALDH1A1 P00352 1/20 0.58
LMNA P02545 1/20 0.58
POLB P06746 1/20 0.58
MAPK1 P28482 1/20 0.58
HSD17B10 Q99714 1/20 0.58
SIGMAR1 Q99720 4/20 0.50
NPSR1 Q6W5P4 1/20 0.50
ABCC1 P33527 2/20 0.49
ABCB1 P08183 1/20 0.49
ABCG2 Q9UNQ0 1/20 0.49
SLC6A3 Q01959 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9683244 0.89 SIGMAR1 (0.54) HTR1ADRD2MAPTALDH1A1LMNA
Hydrochloric Acid SCHEMBL9681380 0.88 SIGMAR1 (0.53) HTR1ADRD2MAPTALDH1A1LMNA
SCHEMBL9681419 0.87 KDM4E (0.49) MAPTALDH1A1LMNAPOLBMAPK1
SCHEMBL9680605 0.87 DRD2 (0.57) HTR1ADRD2MAPTALDH1A1LMNA
SCHEMBL9682450 0.86 DRD4 (0.58) HTR1ADRD2MAPTALDH1A1LMNA
SCHEMBL9680805 0.84 DRD3 (0.43) HTR1ADRD2MAPTALDH1A1LMNA
SCHEMBL9680636 0.83 SMO (0.50) MAPTALDH1A1LMNAMAPK1HSD17B10
SCHEMBL6125292 0.82 KHK (0.56) ALDH1A1
Hydrochloric Acid SCHEMBL9682152 0.81 KHK (0.54) ALDH1A1
SCHEMBL9681924 0.81 HTR1A (0.47) HTR1AMAPTALDH1A1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed