SCHEMBL9682450

SCHEMBL9682450

c1ccc(CN2CCN(c3nn(-c4ccccc4)c4ccccc34)CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.58
LMNA P02545 4/20 0.57
MAPT P10636 2/20 0.57
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
HPGD P15428 1/20 0.57
ACHE P22303 1/20 0.52
HTR3E A5X5Y0 4/20 0.51
HTR3B O95264 4/20 0.51
HTR3A P46098 4/20 0.51
HTR3D Q70Z44 4/20 0.51
HTR3C Q8WXA8 4/20 0.51
HTR1A P08908 2/20 0.51
HTR2C P28335 1/20 0.51
SIGMAR1 Q99720 1/20 0.50
TP53 P04637 1/20 0.48
DRD2 P14416 1/20 0.48
DRD3 P35462 1/20 0.48
KHK P50053 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681250 0.86 HTR1A (0.60) LMNAMAPTALDH1A1HTR1ASIGMAR1
SCHEMBL9680636 0.85 SMO (0.50) LMNAMAPTKDM4EALDH1A1HPGD
SCHEMBL9681419 0.84 KDM4E (0.49) LMNAMAPTKDM4EALDH1A1HTR3E
SCHEMBL9680605 0.84 DRD2 (0.57) LMNAMAPTKDM4EALDH1A1HPGD
SCHEMBL9680621 0.83 KHK (0.44) DRD4LMNAMAPTKDM4EALDH1A1
SCHEMBL9682466 0.83 DRD3 (0.47) DRD4LMNAMAPTKDM4EALDH1A1
SCHEMBL9681924 0.83 HTR1A (0.47) LMNAMAPTKDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL9680620 0.82 HTR1A (0.47) LMNAMAPTKDM4EALDH1A1HPGD
SCHEMBL6125292 0.81 KHK (0.56) KDM4EALDH1A1HTR3EHTR3BHTR3A
SCHEMBL9681353 0.81 KHK (0.42) LMNAMAPTKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed