SCHEMBL9681666

SCHEMBL9681666

CN1C(=O)CC(C)(C)c2cccc([N+](=O)[O-])c21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
TDP1 Q9NUW8 2/20 0.39
GAA P10253 3/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
XDH P47989 1/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
TSHR P16473 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 2/20 0.35
PGR P06401 1/20 0.35
GPR35 Q9HC97 1/20 0.35
S100A4 P26447 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9679997 0.76 BACE1 (0.40) KMT2AMEN1
SCHEMBL9682204 0.72 NOTUM (0.35) ALDH1A1TSHR
SCHEMBL8141328 0.72 ALDH1A1 (0.44) TDP1GAAXDHALDH1A1CYP1A2
SCHEMBL9593368 0.71 ALDH1A1 (0.51) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9378647 0.71 TDP1 (0.41) TDP1KMT2AXDHTSHRSMN1; SMN2
SCHEMBL10442406 0.70 ALDH1A1 (0.42) TDP1GAAKMT2AMEN1XDH
SCHEMBL6748962 0.68 NOTUM (0.45) GAAKMT2AMEN1ALDH1A1TSHR
SCHEMBL5446843 0.67 GABRA1 (0.44) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL2029915 0.67 S100A4 (0.46) TDP1GAAKMT2AXDHALDH1A1
SCHEMBL28281765 0.65 TDP1 (0.41) TDP1GAAKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0504695-A1 New carboxamides, their preparation and pharmaceutical compositions containing them F. HOFFMANN-LA ROCHE AG (CH) 1992-09-23 EP disclosed