SCHEMBL9682204

SCHEMBL9682204

CC(=O)c1cccc2c1N(C)C(=O)CC2(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.35
PDK2 Q15119 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
CBX7 O95931 1/20 0.34
CDY1; CDY1B Q9Y6F8 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
MAP2K1 Q02750 1/20 0.33
KDM4E B2RXH2 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
BRD4 O60885 1/20 0.33
MAP3K5 Q99683 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2230498 0.79 HTR1A (0.36) NOTUMHDAC3HDAC4HDAC1HDAC2
SCHEMBL2231425 0.79 HTR1A (0.36) NOTUMHDAC1HDAC2HDAC6ALDH1A1
SCHEMBL9679997 0.77 BACE1 (0.40) MAP2K1BACE1HTR2AHTR2CHTR2B
SCHEMBL9681666 0.72 GABRA1 (0.39) TSHRALDH1A1
SCHEMBL10559978 0.71 NOTUM (0.44) NOTUMPDK2MAP2K1L3MBTL1
SCHEMBL15135472 0.70 RARB (0.36) NOTUMPDK2HDAC3HDAC4HDAC1
SCHEMBL6748962 0.69 NOTUM (0.45) NOTUMTSHRHTTHDAC3HDAC4
SCHEMBL6770006 0.68 HDAC1 (0.56) HTTHDAC3HDAC4HDAC1HDAC2
SCHEMBL30991208 0.64 PDK2 (0.41) NOTUMPDK2HDAC4KDM4EALDH1A1
SCHEMBL29392112 0.64 ALDH1A1 (0.40) NOTUMPDK2KDM4EL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0504695-A1 New carboxamides, their preparation and pharmaceutical compositions containing them F. HOFFMANN-LA ROCHE AG (CH) 1992-09-23 EP disclosed