SCHEMBL9681760

SCHEMBL9681760

COc1cc(C)c(C)nc1C=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.39
KDM4E B2RXH2 3/20 0.39
TSHR P16473 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
TXNRD1 Q16881 4/20 0.37
TXNRD3 Q86VQ6 4/20 0.37
TXNRD2 Q9NNW7 4/20 0.37
ERN1 O75460 3/20 0.37
PRKDC P78527 2/20 0.36
AOX1 Q06278 1/20 0.34
TRIM24 O15164 1/20 0.34
HPGD P15428 1/20 0.34
ALDH5A1 P51649 1/20 0.34
ABAT P80404 1/20 0.34
TRIM33 Q9UPN9 1/20 0.34
MAPT P10636 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362701 0.79 HMGCR (0.41) ALDH1A1TXNRD1TXNRD3TXNRD2MAPT
SCHEMBL17408855 0.77 BCHE (0.37) ALDH1A1KDM4ETSHRMAPTBCHE
SCHEMBL9846198 0.74 MAPT (0.46) ALDH1A1KDM4EMAPTL3MBTL1ACHE
SCHEMBL20113952 0.74 CYP1A2 (0.39) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL9846087 0.71 ALDH1A1 (0.42) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL9681854 0.69 ALDH1A1 (0.39) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL30705516 0.69 ALDH1A1 (0.39) ALDH1A1KDM4ETSHRTDP1ERN1
SCHEMBL9682798 0.69 TLR8 (0.57) ALDH1A1KDM4EHPGDMAPTACHE
SCHEMBL31353452 0.67 PRKDC (0.39) ALDH1A1KDM4EERN1PRKDCHPGD
SCHEMBL9680324 0.67 NPC1 (0.51) ALDH1A1KDM4ETSHRTDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed