SCHEMBL9681937

SCHEMBL9681937

NC(=O)N1CCN(c2nn(-c3ccccc3)c3cc(F)ccc23)CC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KHK P50053 8/20 0.42
HTR1A P08908 1/20 0.42
HTR2A P28223 1/20 0.42
HTR7 P34969 1/20 0.42
HTR6 P50406 1/20 0.42
LMNA P02545 3/20 0.42
ALDH1A1 P00352 1/20 0.42
RECQL P46063 1/20 0.42
MAP3K14 Q99558 2/20 0.41
PTGER1 P34995 1/20 0.39
MAPT P10636 2/20 0.39
RAB9A P51151 2/20 0.39
SMO Q99835 1/20 0.39
NPC1 O15118 1/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KIT P10721 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680606 0.86 TP53 (0.45) LMNAPTGER1MAPTSMOTSHR
SCHEMBL9681935 0.86 PTGER1 (0.49) KHKHTR1AHTR2AHTR7HTR6
SCHEMBL9680590 0.82 KHK (0.58) KHKMAPTTSHR
Hydrochloric Acid SCHEMBL9682507 0.81 KHK (0.57) KHKHTR6MAPTTSHR
SCHEMBL10395409 0.80 KHK (0.48) KHKMAP3K14
SCHEMBL9681244 0.80 KHK (0.57) KHK
SCHEMBL9763071 0.78 PTGER1 (0.44) HTR1AHTR2AHTR7HTR6LMNA
SCHEMBL9680653 0.77 PTGER1 (0.43) KHKLMNAALDH1A1PTGER1MAPT
SCHEMBL9763297 0.76 SCN9A (0.46) LMNAPTGER1MAPTRAB9ASMN1; SMN2
SCHEMBL9681280 0.74 LMNA (0.45) LMNAALDH1A1PTGER1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed