SCHEMBL9682115

SCHEMBL9682115

CCc1cc(CCc2nc3c(Cl)ccc(Cl)c3o2)c(=S)[nH]c1COCc1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.33
ALDH1A1 P00352 2/20 0.31
CDK5 Q00535 2/20 0.31
CDK5R1 Q15078 2/20 0.31
MEN1 O00255 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
GLA P06280 1/20 0.31
TSHR P16473 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
NPC1 O15118 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
RAB9A P51151 1/20 0.30
MCL1 Q07820 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9682811 0.90 HCAR2 (0.37) HCAR2ALDH1A1CDK5CDK5R1MEN1
SCHEMBL9680858 0.83 ALDH1A1 (0.32) HCAR2ALDH1A1MEN1HPGDKMT2A
SCHEMBL9284917 0.79 ALDH1A1 (0.35) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9682775 0.74 HCAR2 (0.36) HCAR2CDK5CDK5R1
SCHEMBL9682778 0.74 HCAR2 (0.36) HCAR2CDK5CDK5R1
SCHEMBL9601892 0.74 ALDH1A1 (0.36) HCAR2ALDH1A1MEN1HPGDKMT2A
SCHEMBL9449331 0.72 MAPT (0.44) HCAR2CDK5CDK5R1KDM4EMAPT
SCHEMBL9846244 0.67 APOBEC3A (0.30)
SCHEMBL9283236 0.66 ALDH1A1 (0.41) HCAR2ALDH1A1MEN1HPGDKMT2A
SCHEMBL9680279 0.64 TSHR (0.41) HCAR2ALDH1A1CDK5CDK5R1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed