SCHEMBL9601892

SCHEMBL9601892

CCc1cc(CCc2nc3c(Cl)ccc(Cl)c3o2)c(=O)[nH]c1CO

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
HCAR2 Q8TDS4 1/20 0.35
GLA P06280 1/20 0.35
TSHR P16473 1/20 0.35
NPC1 O15118 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
RAB9A P51151 1/20 0.34
MCL1 Q07820 1/20 0.34
HSD17B10 Q99714 1/20 0.34
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
APLNR P35414 1/20 0.30
TYMS P04818 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680858 0.89 ALDH1A1 (0.32) ALDH1A1MEN1HPGDKMT2AHCAR2
SCHEMBL9280809 0.85 ALDH1A1 (0.38) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9680867 0.83 MEN1 (0.36) ALDH1A1MEN1HPGDKMT2AHCAR2
SCHEMBL9682811 0.82 HCAR2 (0.37) ALDH1A1MEN1HPGDKMT2AHCAR2
SCHEMBL9455992 0.82 HCAR2 (0.33) ALDH1A1MEN1HPGDKMT2AHCAR2
SCHEMBL9283236 0.81 ALDH1A1 (0.41) ALDH1A1MEN1HPGDKMT2AHCAR2
SCHEMBL9455991 0.77 HCAR2 (0.34) HCAR2TYMS
SCHEMBL9846309 0.76 FABP4 (0.31) ALDH1A1MEN1HPGDKMT2AHCAR2
SCHEMBL9449230 0.76 MAPT (0.50) MEN1KMT2AHCAR2NPC1RAB9A
SCHEMBL9284917 0.76 ALDH1A1 (0.35) ALDH1A1MEN1HPGDKMT2AGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP claimed
JP-5170740-A None JP disclosed
JP-H05170740-A HYDROXYLATED INHIBITOR OF HIV REVERSE TRANSCRIPTASE MERCK & CO INC 1993-07-09 JP disclosed
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed