SCHEMBL9683390

SCHEMBL9683390

CCCC(NCC(O)COc1ccccc1)(NCC(O)COc1ccccc1)c1ccc(C(N)=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.52
MAPT P10636 2/20 0.48
CASR P41180 3/20 0.44
ADRB2 P07550 4/20 0.44
ADRB1 P08588 4/20 0.44
ADRB3 P13945 4/20 0.44
PARP10 Q53GL7 1/20 0.44
ALDH1A1 P00352 1/20 0.43
ABCB1 P08183 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9684114 0.75 CYP2D6 (0.51) CYP2D6MAPTADRB2ADRB1ADRB3
Benzamide SCHEMBL4775810 0.74 HIF1A (0.58) PARP10ALDH1A1ABCB1
SCHEMBL9812104 0.73 CYP2D6 (0.51) CYP2D6MAPTCASRADRB2ADRB1
SCHEMBL9362874 0.73 CYP2D6 (0.56) CYP2D6MAPTCASRADRB2ADRB1
SCHEMBL9685173 0.71 ADRB1 (0.69) ADRB2ADRB1ADRB3
SCHEMBL9685167 0.71 ADRB1 (0.69) ADRB2ADRB1ADRB3
SCHEMBL9330171 0.71 CYP2D6 (0.58) CYP2D6MAPTCASRADRB2ADRB1
SCHEMBL10822357 0.71 BCAT2 (0.48) MAPTADRB1ADRB3ALDH1A1
SCHEMBL11373388 0.70 CYP2D6 (0.77) CYP2D6MAPTCASRADRB2ADRB1
SCHEMBL9683304 0.70 MEN1 (0.76) CYP2D6ADRB2ADRB1ADRB3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166218-A Antilipemic agents or antiglycemic agents HOFFMANN-LA ROCHE INC. (US) 1992-11-24 US disclosed
US-5064863-A Catabolic activity, obesity, diabetes HOFFMANN-LA ROCHE INC. (US) 1991-11-12 US disclosed
EP-0140243-A2 Phenoxypropanol amines F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1985-05-08 EP disclosed