SCHEMBL9684160

SCHEMBL9684160

CN1C(=O)c2ccc(Cl)cc2C(CC(=O)O)C1=O

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.42
FDFT1 P37268 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
CDC25A P30304 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
WDR5 P61964 1/20 0.38
P2RX7 Q99572 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
FFAR1 O14842 1/20 0.36
MDM2 Q00987 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9685018 0.84 AKR1B1 (0.55) AKR1B1CDC25AMAPTWDR5
SCHEMBL9870877 0.82 ALDH1A1 (0.36) KDM4EHPGDMAPTSMN1; SMN2P2RX7
SCHEMBL9870662 0.79 LMNA (0.39) KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL25876757 0.74 KDM4E (0.43) KDM4EHPGDMAPTSMN1; SMN2FFAR1
SCHEMBL8320575 0.74 ALDH1A1 (0.39) KDM4EHPGDSMN1; SMN2P2RX7CYP11B1
SCHEMBL9870526 0.72 CHRM3 (0.36) KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL11358992 0.71 HSD17B10 (0.47)
SCHEMBL4466269 0.70 MDM2 (0.45) FDFT1KDM4EHPGDCYP11B1CYP11B2
SCHEMBL8727194 0.68 CDC25A (0.63) KDM4EHPGDCDC25AMAPTSMN1; SMN2
SCHEMBL7426387 0.67 ALDH1A1 (0.51) KDM4EHPGDMAPTSMN1; SMN2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5130425-A Antidiabetic agents spiro azetidine-2,4'(1'H)-isoquinoline! 1',3',4(2'H)-triones AMERICAN HOME PRODUCTS CORPORATION (US) 1992-07-14 US disclosed