SCHEMBL9870877

SCHEMBL9870877

COC(=O)NC(=O)CC1C(=O)N(C)C(=O)c2ccc(Cl)cc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
HPGD P15428 3/20 0.36
MAPT P10636 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
P2RX7 Q99572 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
POLB P06746 2/20 0.34
CDYL2 Q8N8U2 1/20 0.34
CDYL Q9Y232 1/20 0.34
PTGDR Q13258 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
TSHR P16473 1/20 0.34
GAA P10253 1/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870526 0.91 CHRM3 (0.36) ALDH1A1KDM4ESMN1; SMN2HPGDMAPT
SCHEMBL9870662 0.90 LMNA (0.39) ALDH1A1KDM4ESMN1; SMN2HPGDMAPT
SCHEMBL9871624 0.83 ALDH1A1 (0.38) ALDH1A1KDM4ESMN1; SMN2HPGDCYP3A4
SCHEMBL9684160 0.82 AKR1B1 (0.42) KDM4ESMN1; SMN2HPGDMAPTP2RX7
SCHEMBL8320575 0.75 ALDH1A1 (0.39) ALDH1A1KDM4ESMN1; SMN2HPGDNPSR1
SCHEMBL9384033 0.68 ALDH1A1 (0.41) ALDH1A1KDM4ESMN1; SMN2HPGDCYP2C9
SCHEMBL11788765 0.61 KDM4E (0.38) ALDH1A1KDM4ESMN1; SMN2HPGDCYP2C9
SCHEMBL8322814 0.60 TDP2 (0.47) ALDH1A1SMN1; SMN2CYP2C9CYP2C19NPSR1
SCHEMBL16269466 0.60 CYP11B1 (0.52) P2RX7
SCHEMBL8993321 0.60 HTR2B (0.40) ALDH1A1SMN1; SMN2HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4983613-A Acetamides; treatment of neuropathy, nephropathy, retinopathy or cataracts in diabetic mammals AMERICAN HOME PRODUCTS CORPORATION (US) 1991-01-08 US claimed
US-4983613-A Acetamides; treatment of neuropathy, nephropathy, retinopathy or cataracts in diabetic mammals AMERICAN HOME PRODUCTS CORPORATION (US) 1991-01-08 US disclosed