SCHEMBL9684182

SCHEMBL9684182

Cc1ccc(-c2ccc3c(c2)C=NCC(=O)N3)n1Cl

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PGR P06401 4/20 0.36
NR3C2 P08235 4/20 0.33
NR3C1 P04150 1/20 0.32
PDE4D Q08499 2/20 0.31
CNR1 P21554 1/20 0.31
NTSR1 P30989 1/20 0.31
OPRK1 P41145 1/20 0.31
GRIA1 P42261 2/20 0.31
CACNG8 Q8WXS5 2/20 0.31
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
MMP12 P39900 1/20 0.30
RAB9A P51151 1/20 0.30
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11412815 0.72 AHR (0.49) PGRPDE4DCNR1NTSR1OPRK1
SCHEMBL613060 0.65 GABRA1 (0.44) PDE4DCNR1NTSR1OPRK1NPC1
SCHEMBL4596854 0.63 KIF11 (0.47) GRIA1PDE3BPDE3A
SCHEMBL30908764 0.61 PGR (0.36) PGRPDE4DCNR1NTSR1OPRK1
SCHEMBL10373736 0.59 GABRA1 (0.30)
SCHEMBL30908740 0.58 CES1 (0.39) PGRPDE4DCNR1NTSR1OPRK1
SCHEMBL18322204 0.56 GABRA1 (0.33) MAPT
SCHEMBL1460212 0.55 PGR (0.55) PGRPDE4DGRIA1CACNG8PDE3B
SCHEMBL2464690 0.54
SCHEMBL4435837 0.54 ALDH1A1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0491218-A1 Benzodiazepinones F. HOFFMANN-LA ROCHE AG (CH) 1992-06-24 EP claimed
EP-0491218-A1 Benzodiazepinones F. HOFFMANN-LA ROCHE AG (CH) 1992-06-24 EP disclosed